THE SYNTHESIS OF 2-SUBSTITUTED-1,4-DIHYDROPYRIDINES

被引：8

作者：

ALKER, D

DENTON, SM

机构：

[1] Pfizer Central Research, Sandwich

来源：

TETRAHEDRON | 1990年 / 46卷 / 10期

关键词：

D O I：

10.1016/S0040-4020(01)81539-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reaction of the 2-hydroxymethyl-1,4-dihydropyridines 7 and 13 with SO2Cl2limidazole followed by treatment with nucleophiles affords 2-substituted-l,4-dihydropyridines via the intermediacy of the 2-chloromethyl compounds 14 and 18, respectively. © 1990.

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页码：3693 / 3702

页数：10

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