INDUCTION OF DRUG-METABOLIZING-ENZYMES BY TRICYCLIC ANTI-DEPRESSANTS IN HUMAN-LIVER - CHARACTERIZATION AND PARTIAL RESOLUTION OF CYTOCHROMES P-450

被引:16
作者
CRESTEIL, T [1 ]
CELIER, C [1 ]
KREMERS, P [1 ]
FLINOIS, JP [1 ]
BEAUNE, P [1 ]
LEROUX, JP [1 ]
机构
[1] UNIV LIEGE, INST PATHOL, CHIME MED LAB, B-4000 LIEGE, BELGIUM
关键词
D O I
10.1111/j.1365-2125.1983.tb02236.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:651 / 657
页数:7
相关论文
共 48 条
  • [1] SIMPLE AND SENSITIVE ASSAY OF 7-ETHOXYCOUMARIN DEETHYLATION
    AITIO, A
    [J]. ANALYTICAL BIOCHEMISTRY, 1978, 85 (02) : 488 - 491
  • [2] PARTIAL-PURIFICATION OF HUMAN-LIVER CYTOCHROME-P-450
    BEAUNE, P
    DANSETTE, P
    FLINOIS, JP
    COLUMELLI, S
    MANSUY, D
    LEROUX, JP
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 88 (03) : 826 - 832
  • [3] BEAUNE P, 1980, MICROSOMES DRUG OXID, P107
  • [4] BLACK M, 1973, J LAB CLIN MED, V81, P704
  • [5] EFFECT OF RIFAMPICIN TREATMENT ON METABOLISM OF ESTRADIOL AND 17 ALPHA-ETHINYLESTRADIOL BY HUMAN LIVER-MICROSOMES
    BOLT, HM
    KAPPUS, H
    BOLT, M
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1975, 8 (05) : 301 - 307
  • [6] MONO-OXYGENASE ACTIVITY OF HUMAN-LIVER IN MICROSOMAL FRACTIONS OF NEEDLE-BIOPSY SPECIMENS
    BOOBIS, AR
    BRODIE, MJ
    KAHN, GC
    FLETCHER, DR
    SAUNDERS, JH
    DAVIES, DS
    [J]. BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 9 (01) : 11 - 19
  • [7] CONNEY AH, 1967, PHARMACOL REV, V19, P317
  • [8] CONNEY AH, 1956, CANCER RES, V16, P450
  • [9] Coon M J, 1978, Methods Enzymol, V52, P109
  • [10] CRESTEIL T, 1982, PEDIATR PHARMACOL, V2, P199