SYNTHESIS OF PEPTIDES RELATED TO THE PROSEGMENT OF MOUSE SUBMAXILLARY-GLAND RENIN PRECURSOR - AN APPROACH TO RENIN INHIBITORS

被引:41
作者
EVIN, G [1 ]
DEVIN, J [1 ]
CASTRO, B [1 ]
MENARD, J [1 ]
CORVOL, P [1 ]
机构
[1] CTR PHARMACOL ENDOCRINOL,CNRS,INSERM,F-34033 MONTPELLIER,FRANCE
来源
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES | 1984年 / 81卷 / 01期
关键词
D O I
10.1073/pnas.81.1.48
中图分类号
Q [生物科学];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:48 / 52
页数:5
相关论文
共 38 条
[1]  
ANWER MK, 1980, SYNTHESIS-STUTTGART, V11, P929
[2]   NEW PEPSTATINS, PEPSTATINS BU, PR AND AC PRODUCED BY STREPTOMYCES [J].
AOYAGI, T ;
YAGISAWA, Y ;
KUMAGAI, M ;
HAMADA, M ;
MORISHIMA, H ;
TAKEUCHI, T ;
UMEZAWA, H .
JOURNAL OF ANTIBIOTICS, 1973, 26 (09) :539-541
[3]   EFFECT OF PEPSTATIN ON ACID PROTEASES [J].
AOYAGI, T ;
KUNIMOTO, S ;
MORISHIMA, H ;
TAKEUCHI, T ;
UMEZAWA, H .
JOURNAL OF ANTIBIOTICS, 1971, 24 (10) :687-+
[4]  
ATLAS SA, 1982, HYPERTENSION DALL S2, V4, P87
[5]   NOVEL RENIN INHIBITORS CONTAINING THE AMINO-ACID STATINE [J].
BOGER, J ;
LOHR, NS ;
ULM, EH ;
POE, M ;
BLAINE, EH ;
FANELLI, GM ;
LIN, TY ;
PAYNE, LS ;
SCHORN, TW ;
LAMONT, BI ;
VASSIL, TC ;
STABILITO, II ;
VEBER, DF ;
RICH, DH ;
BOPARI, AS .
NATURE, 1983, 303 (5912) :81-84
[6]   COMPETITIVE INHIBITORS OF RENIN INHIBITORS EFFECTIVE AT PHYSIOLOGICAL PH [J].
BURTON, J ;
POULSEN, K ;
HABER, E .
BIOCHEMISTRY, 1975, 14 (17) :3892-3898
[7]  
CASTRO B, 1975, TETRAHEDRON LETT, P1219
[8]   A SUBSTRATE-ANALOG INHIBITOR OF RENIN THAT IS EFFECTIVE INVIVO [J].
CODY, RJ ;
BURTON, J ;
EVIN, G ;
POULSEN, K ;
HERD, JA ;
HABER, E .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 97 (01) :230-235
[9]   SIMPLE GRAPHICAL METHOD FOR DETERMINING INHIBITION CONSTANTS OF MIXED, UNCOMPETITIVE AND NON-COMPETITIVE INHIBITORS [J].
CORNISHB.A .
BIOCHEMICAL JOURNAL, 1974, 137 (01) :143-144
[10]  
DUNN BM, 1978, J BIOL CHEM, V253, P7269