ASYMMETRIC SYNTHESES VIA HETEROCYCLIC INTERMEDIATES .32. ASYMMETRIC-SYNTHESIS OF CYCLIC ALPHA-AMINO-ACIDS BY THE BISLACTIM ETHER METHOD

被引：62

作者：

SCHOLLKOPF, U

HINRICHS, R

LONSKY, R

机构：

来源：

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION | 1987年 / 26卷 / 02期

关键词：

D O I：

10.1002/anie.198701431

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Methylproline, 1a, and its cyclic homologues, 1b and 2, have been synthesized without direct recourse to the "chiral pool". The multistep synthesis starts from the bislactim either 3 and the dibromides 4a,b and 5 (a, n=1; b, n=2).

引用

页码：143 / 145

页数：3

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[3]

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[7]

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