HIGH AND LOW (GPP(NH)P-SENSITIVE) AFFINITY SITES FOR BETA-2-ADRENERGIC BLOCKERS AS ANTAGONISTS OF ISOPROTERENOL IN THE FIELD-STIMULATED RAT VAS-DEFERENS

被引:7
作者
LOTTI, VJ [1 ]
KLING, P [1 ]
CERINO, D [1 ]
机构
[1] MERCK INST THERAPEUT RES,MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
关键词
D O I
10.1016/0014-2999(82)90198-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
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页码:161 / 167
页数:7
相关论文
共 17 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]   ADRENERGIC NEURON BLOCKING PROPERTIES OF (+/-)-PROPRANOLOL AND (+)-PROPRANOLOL [J].
BARRETT, AM ;
NUNN, B .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1970, 22 (11) :806-+
[3]   COMPARISON OF PHARMACOLOGICAL AND BINDING ASSAYS FOR 10 BETA-ADRENOCEPTOR BLOCKING-AGENTS AND 2 BETA-ADRENOCEPTOR AGONISTS [J].
BIETH, N ;
ROUOT, B ;
SCHWARTZ, J ;
VELLY, J .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 68 (03) :563-569
[4]   EFFECTS OF ALPHA-ADRENOCEPTOR AGONISTS AND ANTAGONISTS ON RESPONSES OF TRANSMURALLY STIMULATED PROSTATIC AND EPIDIDYMAL PORTIONS OF THE ISOLATED VAS-DEFERENS OF THE RAT [J].
BROWN, CM ;
MCGRATH, JC ;
SUMMERS, RJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1979, 66 (04) :553-564
[5]  
DALY MJ, 1979, TRENDS AUTONOMIC PHA, V1, P347
[6]   SELECTIVITY OF BLOCKING-AGENTS FOR PRESYNAPTIC AND POSTSYNAPTIC ALPHA-ADRENOCEPTORS [J].
DOXEY, JC ;
SMITH, CFC ;
WALKER, JM .
BRITISH JOURNAL OF PHARMACOLOGY, 1977, 60 (01) :91-96
[7]   PHARMACOLOGICAL CHARACTERIZATION OF PRESYNAPTIC ALPHA-ADRENOCEPTOR IN RAT VAS-DEFERENS [J].
DREW, GM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1977, 42 (02) :123-130
[8]   INVESTIGATIONS ON THE MODE OF ACTION OF A NEW ANTIHYPERTENSIVE DRUG, URAPIDIL, IN THE ISOLATED RAT VAS-DEFERENS [J].
ELTZE, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 59 (1-2) :1-9
[9]   RADIOLIGAND BINDING-STUDIES OF ADRENERGIC-RECEPTORS - NEW INSIGHTS INTO MOLECULAR AND PHYSIOLOGICAL REGULATION [J].
HOFFMAN, BB ;
LEFKOWITZ, RJ .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1980, 20 :581-608
[10]   POTENT NEW BETA2-ADRENOCEPTOR BLOCKING-AGENT [J].
IMBS, JL ;
MIESCH, F ;
SCHWARTZ, J ;
VELLY, J ;
LECLERC, G ;
MANN, A ;
WERMUTH, CG .
BRITISH JOURNAL OF PHARMACOLOGY, 1977, 60 (03) :357-362