N-T-BUTOXYCARBONYL PROTECTION OF PRIMARY AND SECONDARY-AMINES IN THE HYDROBORATION REACTION - SYNTHESIS OF AMINO-ALCOHOLS

被引：11

作者：

KABALKA, GW ^{[1
]}

LI, NS ^{[1
]}

PACE, RD ^{[1
]}

机构：

[1] UNIV TENNESSEE,DEPT RADIOL,KNOXVILLE,TN 37996

来源：

SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 14期

关键词：

D O I：

10.1080/00397919508015894

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The use of the BOC group as a protecting group in the hydroboration of aminoalkenes is described. The isolated yields of amino alcohols via the hydroboration-oxidation sequence are excellent.

引用

页码：2135 / 2143

页数：9

共 33 条

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