TITANIUM(IV) MEDIATED REDUCTIVE AMINATIONS OF 1-ADAMANTYL METHYL KETONE - FACILE PREPARATION OF POTENTIAL ANTIVIRAL AGENTS RIMANTADINE AND ITS ANALOGS

被引：12

作者：

BHATTACHARYYA, S ^{[1
]}

机构：

[1] VIJOYGARH COLL,DEPT CHEM,CALCUTTA 700032,W BENGAL,INDIA

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1995年 / 14期

关键词：

D O I：

10.1039/p19950001845

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A preparatively efficient, mild method for the synthesis of rimantadine and its analogues via novel reductive aminations of l-adamantyl methyl ketone using titanium(IV) isopropoxide and sodium borohydride is reported.

引用

页码：1845 / 1847

页数：3

共 29 条

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