POLYMER-BOUND EDC (P-EDC) - A CONVENIENT REAGENT FOR FORMATION OF AN AMIDE BOND

被引：124

作者：

DESAI, MC

STRAMIELLO, LMS

机构：

[1] Central Research Division, Pfizer Inc., Groton

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 48期

关键词：

D O I：

10.1016/S0040-4039(00)61539-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A facile preparation of polymer bound 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide (P-EDC) from commercially available starting materials is described. The P-EDC was found to be a convenient and general reagent for coupling of a variety of amines with diverse carboxylic acids.

引用

页码：7685 / 7688

页数：4

共 22 条

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