共 15 条
[5]
TUMOR GROWTH-STIMULATING AND INHIBITING EFFECTS OF ANTI-ESTROGENS ON THE DMBA-INDUCED MAMMARY-CARCINOMA OF THE OVARIECTOMIZED, DIETHYLSTILBESTROL-TREATED SD RAT - A STUDY ON THE MECHANISM OF ACTION OF ANTI-ESTROGENS
[J].
EUROPEAN JOURNAL OF CANCER & CLINICAL ONCOLOGY,
1983, 19 (07)
:959-964
[7]
RING-SUBSTITUTED 1,2-DIALKYLATED 1,2-BIS(HYDROXYPHENYL)ETHANES .3. SYNTHESIS, ESTROGEN-RECEPTOR BINDING-AFFINITY, AND EVALUATION OF ANTIESTROGENIC AND MAMMARY-TUMOR INHIBITING ACTIVITY OF 2,2'-DISUBSTITUTED BUTESTROLS AND 6,6'-DISUBSTITUTED METABUTESTROLS
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1984, 27 (07)
:819-824
[9]
HARTMANN RW, 1985, J MED CHEM, V10, P48
[10]
ANTIESTROGENS .2. STRUCTURE ACTIVITY STUDIES IN A SERIES OF 3-AROYL-2-ARYLBENZO[B]THIOPHENE DERIVATIVES LEADING TO [6-HYDROXY-2-(4-HYDROXYPHENYL)BENZO[B]THIEN-3-YL][4-[2-(1-PIPERIDINYL)ETHOXY]-PHENYL]METHANONE HYDROCHLORIDE (LY156758), A REMARKABLY EFFECTIVE ESTROGEN ANTAGONIST WITH ONLY MINIMAL INTRINSIC ESTROGENICITYO[
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1984, 27 (08)
:1057-1066