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L-656,224 (7-CHLORO-2-[(4-METHOXYPHENYL)METHYL]-3-METHYL-5-PROPYL-4-BENZOFURANOL) - A NOVEL, SELECTIVE, ORALLY ACTIVE 5-LIPOXYGENASE INHIBITOR
被引:33
作者
:
BELANGER, P
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
BELANGER, P
MAYCOCK, A
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
MAYCOCK, A
GUINDON, Y
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
GUINDON, Y
BACH, T
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
BACH, T
DOLLOB, AL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
DOLLOB, AL
DUFRESNE, C
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
DUFRESNE, C
FORDHUTCHINSON, AW
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
FORDHUTCHINSON, AW
GALE, PH
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
GALE, PH
HOPPLE, S
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
HOPPLE, S
LAU, CK
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
LAU, CK
LETTS, LG
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
LETTS, LG
LUELL, S
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
LUELL, S
MCFARLANE, CS
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
MCFARLANE, CS
MACINTYRE, E
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
MACINTYRE, E
MEURER, R
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
MEURER, R
MILLER, DK
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
MILLER, DK
PIECHUTA, H
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
PIECHUTA, H
RIENDEAU, D
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
RIENDEAU, D
ROKACH, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
ROKACH, J
ROUZER, C
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
ROUZER, C
SCHEIGETZ, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
SCHEIGETZ, J
机构
:
[1]
MERCK FROSST CANADA INC,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
[2]
MERCK FROSST CANADA INC,DEPT PHARMACOL,MONTREAL,QUEBEC,CANADA
[3]
MERCK FROSST CANADA INC,DEPT MED CHEM,MONTREAL,QUEBEC,CANADA
[4]
MERCK SHARP & DOHME RES LABS,DEPT BIOCHEM & INFLAMMAT,RAHWAY,NJ 07065
[5]
MERCK FROSST CANADA INC,DEPT PHARMACOL & MED CHEM,MONTREAL,QUEBEC,CANADA
来源
:
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY
|
1987年
/ 65卷
/ 12期
关键词
:
D O I
:
10.1139/y87-387
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
引用
收藏
页码:2441 / 2448
页数:8
相关论文
共 24 条
[1]
MEASUREMENT OF CUTANEOUS INFLAMMATION - ESTIMATION OF NEUTROPHIL CONTENT WITH AN ENZYME MARKER
BRADLEY, PP
论文数:
0
引用数:
0
h-index:
0
BRADLEY, PP
PRIEBAT, DA
论文数:
0
引用数:
0
h-index:
0
PRIEBAT, DA
CHRISTENSEN, RD
论文数:
0
引用数:
0
h-index:
0
CHRISTENSEN, RD
ROTHSTEIN, G
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0
引用数:
0
h-index:
0
ROTHSTEIN, G
[J].
JOURNAL OF INVESTIGATIVE DERMATOLOGY,
1982,
78
(03)
: 206
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209
[2]
BRUNET G, 1983, J IMMUNOL, V131, P434
[3]
PHARMACOLOGICAL EVIDENCE FOR A ROLE OF LIPOXYGENASE PRODUCTS IN PLATELET-ACTIVATING-FACTOR (PAF)-INDUCED HYPERALGESIA
DALLOB, A
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
DALLOB, A
GUINDON, Y
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
GUINDON, Y
GOLDENBERG, MM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
GOLDENBERG, MM
[J].
BIOCHEMICAL PHARMACOLOGY,
1987,
36
(19)
: 3201
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3204
[4]
EGAN RW, 1976, J BIOL CHEM, V251, P7329
[5]
EGAN RW, 1985, J BIOL CHEM, V260, P1554
[6]
LEUKOTRIENE-B, A POTENT CHEMOKINETIC AND AGGREGATING SUBSTANCE RELEASED FROM POLYMORPHONUCLEAR LEUKOCYTES
FORDHUTCHINSON, AW
论文数:
0
引用数:
0
h-index:
0
FORDHUTCHINSON, AW
BRAY, MA
论文数:
0
引用数:
0
h-index:
0
BRAY, MA
DOIG, MV
论文数:
0
引用数:
0
h-index:
0
DOIG, MV
SHIPLEY, ME
论文数:
0
引用数:
0
h-index:
0
SHIPLEY, ME
SMITH, MJH
论文数:
0
引用数:
0
h-index:
0
SMITH, MJH
[J].
NATURE,
1980,
286
(5770)
: 264
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265
[7]
LATE PULMONARY RESPONSES INDUCED BY ASCARIS ALLERGEN IN CONSCIOUS SQUIRREL-MONKEYS
HAMEL, R
论文数:
0
引用数:
0
h-index:
0
HAMEL, R
MCFARLANE, CS
论文数:
0
引用数:
0
h-index:
0
MCFARLANE, CS
FORDHUTCHINSON, AW
论文数:
0
引用数:
0
h-index:
0
FORDHUTCHINSON, AW
[J].
JOURNAL OF APPLIED PHYSIOLOGY,
1986,
61
(06)
: 2081
-
2087
[8]
LETTS LG, 1987, ADV PROSTAGLANDIN TH, V17, P1003
[9]
LEUKOTRIENE-B4 PRODUCES HYPERALGESIA THAT IS DEPENDENT ON POLYMORPHONUCLEAR LEUKOCYTES
LEVINE, JD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
LEVINE, JD
LAU, W
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
LAU, W
KWIAT, G
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
KWIAT, G
GOETZL, EJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
GOETZL, EJ
[J].
SCIENCE,
1984,
225
(4663)
: 743
-
745
[10]
EFFECTS OF A CONTRACTILE PROSTAGLANDIN ANTAGONIST (L-640,035) UPON ALLERGEN-INDUCED BRONCHOCONSTRICTION IN HYPERREACTIVE RATS AND CONSCIOUS SQUIRREL-MONKEYS
MCFARLANE, CS
论文数:
0
引用数:
0
h-index:
0
MCFARLANE, CS
PIECHUTA, H
论文数:
0
引用数:
0
h-index:
0
PIECHUTA, H
HALL, RA
论文数:
0
引用数:
0
h-index:
0
HALL, RA
FORDHUTCHINSON, AW
论文数:
0
引用数:
0
h-index:
0
FORDHUTCHINSON, AW
[J].
PROSTAGLANDINS & OTHER LIPID MEDIATORS,
1984,
28
(02)
: 173
-
182
←
1
2
3
→
共 24 条
[1]
MEASUREMENT OF CUTANEOUS INFLAMMATION - ESTIMATION OF NEUTROPHIL CONTENT WITH AN ENZYME MARKER
BRADLEY, PP
论文数:
0
引用数:
0
h-index:
0
BRADLEY, PP
PRIEBAT, DA
论文数:
0
引用数:
0
h-index:
0
PRIEBAT, DA
CHRISTENSEN, RD
论文数:
0
引用数:
0
h-index:
0
CHRISTENSEN, RD
ROTHSTEIN, G
论文数:
0
引用数:
0
h-index:
0
ROTHSTEIN, G
[J].
JOURNAL OF INVESTIGATIVE DERMATOLOGY,
1982,
78
(03)
: 206
-
209
[2]
BRUNET G, 1983, J IMMUNOL, V131, P434
[3]
PHARMACOLOGICAL EVIDENCE FOR A ROLE OF LIPOXYGENASE PRODUCTS IN PLATELET-ACTIVATING-FACTOR (PAF)-INDUCED HYPERALGESIA
DALLOB, A
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
DALLOB, A
GUINDON, Y
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
GUINDON, Y
GOLDENBERG, MM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
MERCK FROSST CANADA,QUEBEC CITY H9R 4P8,QUEBEC,CANADA
GOLDENBERG, MM
[J].
BIOCHEMICAL PHARMACOLOGY,
1987,
36
(19)
: 3201
-
3204
[4]
EGAN RW, 1976, J BIOL CHEM, V251, P7329
[5]
EGAN RW, 1985, J BIOL CHEM, V260, P1554
[6]
LEUKOTRIENE-B, A POTENT CHEMOKINETIC AND AGGREGATING SUBSTANCE RELEASED FROM POLYMORPHONUCLEAR LEUKOCYTES
FORDHUTCHINSON, AW
论文数:
0
引用数:
0
h-index:
0
FORDHUTCHINSON, AW
BRAY, MA
论文数:
0
引用数:
0
h-index:
0
BRAY, MA
DOIG, MV
论文数:
0
引用数:
0
h-index:
0
DOIG, MV
SHIPLEY, ME
论文数:
0
引用数:
0
h-index:
0
SHIPLEY, ME
SMITH, MJH
论文数:
0
引用数:
0
h-index:
0
SMITH, MJH
[J].
NATURE,
1980,
286
(5770)
: 264
-
265
[7]
LATE PULMONARY RESPONSES INDUCED BY ASCARIS ALLERGEN IN CONSCIOUS SQUIRREL-MONKEYS
HAMEL, R
论文数:
0
引用数:
0
h-index:
0
HAMEL, R
MCFARLANE, CS
论文数:
0
引用数:
0
h-index:
0
MCFARLANE, CS
FORDHUTCHINSON, AW
论文数:
0
引用数:
0
h-index:
0
FORDHUTCHINSON, AW
[J].
JOURNAL OF APPLIED PHYSIOLOGY,
1986,
61
(06)
: 2081
-
2087
[8]
LETTS LG, 1987, ADV PROSTAGLANDIN TH, V17, P1003
[9]
LEUKOTRIENE-B4 PRODUCES HYPERALGESIA THAT IS DEPENDENT ON POLYMORPHONUCLEAR LEUKOCYTES
LEVINE, JD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
LEVINE, JD
LAU, W
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
LAU, W
KWIAT, G
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
KWIAT, G
GOETZL, EJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,DEPT MED,DIV ORAL & MAXILLOFACIAL SURG,SAN FRANCISCO,CA 94143
GOETZL, EJ
[J].
SCIENCE,
1984,
225
(4663)
: 743
-
745
[10]
EFFECTS OF A CONTRACTILE PROSTAGLANDIN ANTAGONIST (L-640,035) UPON ALLERGEN-INDUCED BRONCHOCONSTRICTION IN HYPERREACTIVE RATS AND CONSCIOUS SQUIRREL-MONKEYS
MCFARLANE, CS
论文数:
0
引用数:
0
h-index:
0
MCFARLANE, CS
PIECHUTA, H
论文数:
0
引用数:
0
h-index:
0
PIECHUTA, H
HALL, RA
论文数:
0
引用数:
0
h-index:
0
HALL, RA
FORDHUTCHINSON, AW
论文数:
0
引用数:
0
h-index:
0
FORDHUTCHINSON, AW
[J].
PROSTAGLANDINS & OTHER LIPID MEDIATORS,
1984,
28
(02)
: 173
-
182
←
1
2
3
→