N-(3-ACETYLAMINOPHENYL)PIPERAZINE HYDROCHLORIDE (BEA-1654), A PUTATIVE 5-HT1 AGONIST, CAUSES CONSTRICTION OF ARTERIOVENOUS ANASTOMOSES AND DILATATION OF ARTERIOLES

被引:23
作者
VERDOUW, PD
JENNEWEIN, HM
MIERAU, J
SAXENA, PR
机构
[1] ERASMUS UNIV,DEPT PHARMACOL,3000 DR ROTTERDAM,NETHERLANDS
[2] BOEHRINGER INGELHEIM KG,INGELHEIM,FED REP GER
关键词
D O I
10.1016/0014-2999(85)90259-6
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:337 / 346
页数:10
相关论文
共 27 条
[1]   EVIDENCE FOR 2 TYPES OF EXCITATORY RECEPTOR FOR 5-HYDROXYTRYPTAMINE IN DOG ISOLATED VASCULATURE [J].
APPERLEY, E ;
FENIUK, W ;
HUMPHREY, PPA ;
LEVY, GP .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 68 (02) :215-224
[2]  
BENNETT JP, 1976, MOL PHARMACOL, V12, P373
[3]   OPERATIONAL MODELS OF PHARMACOLOGICAL AGONISM [J].
BLACK, JW ;
LEFF, P .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1983, 220 (1219) :141-162
[4]  
DESHMUKH PP, 1982, FED PROC, V41, P6238
[5]   EVIDENCE FOR COMMON PHARMACOLOGICAL PROPERTIES OF [H-3]5-HYDROXYTRYPTAMINE BINDING-SITES, PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE AUTORECEPTORS IN CNS AND INHIBITORY PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE RECEPTORS ON SYMPATHETIC-NERVES [J].
ENGEL, G ;
GOTHERT, M ;
MULLERSCHWEINITZER, E ;
SCHLICKER, E ;
SISTONEN, L ;
STADLER, PA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 324 (02) :116-124
[7]   BINDING CHARACTERISTICS OF PRAZOSIN-H-3 TO RAT-BRAIN ALPHA-ADRENERGIC RECEPTORS [J].
GREENGRASS, P ;
BREMNER, R .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 55 (03) :323-326
[8]  
JENNEWEIN H M, 1984, British Journal of Pharmacology, V82, p208P
[9]   EFFECT OF ERGOTAMINE ON TISSUE BLOOD-FLOW AND ARTERIOVENOUS SHUNTING OF RADIOACTIVE MICROSPHERES IN HEAD [J].
JOHNSTON, BM ;
SAXENA, PR .
BRITISH JOURNAL OF PHARMACOLOGY, 1978, 63 (03) :541-549
[10]  
KALKMAN HO, 1983, THESIS U AMSTERDAM N