COMPARATIVE-ANALYSIS OF 2 TYPES OF 5-HYDROXYTRYPTAMINE RECEPTOR MEDIATING VASORELAXATION - DIFFERENTIAL CLASSIFICATION USING TRYPTAMINES

被引:65
作者
MARTIN, GR
LEFF, P
CAMBRIDGE, D
BARRETT, VJ
机构
关键词
D O I
10.1007/BF00164867
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:365 / 373
页数:9
相关论文
共 36 条
[1]   PHARMACOLOGICAL ANALYSIS OF THE INTERACTION BETWEEN BAY-K 8644 AND 5-HT IN RABBIT AORTA [J].
BARRETT, VJ ;
LEFF, P ;
MARTIN, GR ;
RICHARDSON, PJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 87 (03) :487-494
[2]   OPERATIONAL MODELS OF PHARMACOLOGICAL AGONISM [J].
BLACK, JW ;
LEFF, P .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1983, 220 (1219) :141-162
[3]   AN OPERATIONAL MODEL OF PHARMACOLOGICAL AGONISM - THE EFFECT OF E/[A] CURVE SHAPE ON AGONIST DISSOCIATION-CONSTANT ESTIMATION [J].
BLACK, JW ;
LEFF, P ;
SHANKLEY, NP ;
WOOD, J .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (02) :561-571
[4]   PROPOSALS FOR THE CLASSIFICATION AND NOMENCLATURE OF FUNCTIONAL RECEPTORS FOR 5-HYDROXYTRYPTAMINE [J].
BRADLEY, PB ;
ENGEL, G ;
FENIUK, W ;
FOZARD, JR ;
HUMPHREY, PPA ;
MIDDLEMISS, DN ;
MYLECHARANE, EJ ;
RICHARDSON, BP ;
SAXENA, PR .
NEUROPHARMACOLOGY, 1986, 25 (06) :563-576
[5]  
BUCHHEIT K H, 1986, British Journal of Pharmacology, V88, p367P
[6]  
CLANCY BM, 1985, J PHARMACOL EXP THER, V233, P761
[7]   ENDOTHELIUM-DEPENDENT RELAXATION OF CORONARY-ARTERIES BY NORADRENALINE AND SEROTONIN [J].
COCKS, TM ;
ANGUS, JA .
NATURE, 1983, 305 (5935) :627-630
[8]   5-CARBOXAMIDOTRYPTAMINE IS A SELECTIVE AGONIST AT 5-HYDROXYTRYPTAMINE RECEPTORS MEDIATING VASODILATATION AND TACHYCARDIA IN ANESTHETIZED CATS [J].
CONNOR, HE ;
FENIUK, W ;
HUMPHREY, PPA ;
PERREN, MJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 87 (02) :417-426
[9]   AN INVESTIGATION INTO THE MECHANISMS OF THE CARDIOVASCULAR EFFECTS OF 5-HYDROXYTRYPTAMINE IN CONSCIOUS NORMOTENSIVE AND DOCA-SALT HYPERTENSIVE RATS [J].
DALTON, DW ;
FENIUK, W ;
HUMPHREY, PPA .
JOURNAL OF AUTONOMIC PHARMACOLOGY, 1986, 6 (03) :219-228
[10]   SEROTONIN INCREASES THE PRODUCTION OF INOSITOL PHOSPHATES AND MOBILIZES CALCIUM VIA THE 5-HT2 RECEPTOR IN A7R5 SMOOTH-MUSCLE CELLS [J].
DOYLE, VM ;
CREBA, JA ;
RUEGG, UT ;
HOYER, D .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1986, 333 (02) :98-103