EXVIVO INHIBITION OF RAT-BRAIN CYTOCHROME-P-450 ACTIVITY BY STIRIPENTOL

被引:15
作者
MESNIL, M
TESTA, B
JENNER, P
机构
[1] UNIV LAUSANNE,SCH PHARM,PL CHATEAU,CH-1005 LAUSANNE,SWITZERLAND
[2] UNIV LONDON,INST PSYCHIAT,DEPT NEUROL,LONDON SE5 8AF,ENGLAND
[3] UNIV LONDON KINGS COLL HOSP,SCH MED,LONDON SE5 8AF,ENGLAND
关键词
D O I
10.1016/0006-2952(88)90393-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3619 / 3622
页数:4
相关论文
共 14 条
[1]   LIGAND-COMPLEX FORMATION BETWEEN CYTOCHROME-P-450 AND CYTOCHROME-P448 AND METHYLENEDIOXYPHENYL COMPOUNDS [J].
DELAFORGE, M ;
IOANNIDES, C ;
PARKE, DV .
XENOBIOTICA, 1985, 15 (04) :333-342
[2]   STIRIPENTOL KINETICS IN EPILEPSY - NONLINEARITY AND INTERACTIONS [J].
LEVY, RH ;
LOISEAU, P ;
GUYOT, M ;
BLEHAUT, HM ;
TOR, J ;
MORELAND, TA .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1984, 36 (05) :661-669
[3]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265
[4]   SPECTRAL AND INHIBITORY INTERACTIONS OF METHYLENEDIOXYPHENYL AND RELATED-COMPOUNDS WITH PURIFIED ISOZYMES OF CYTOCHROME-P-450 [J].
MARCUS, CB ;
MURRAY, M ;
WILKINSON, CF .
XENOBIOTICA, 1985, 15 (04) :351-362
[5]   ARYL-HYDROCARBON HYDROXYLASE IN RAT-BRAIN MICROSOMES [J].
MESNIL, M ;
TESTA, B ;
JENNER, P .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (03) :435-436
[6]  
Mesnil M., 1984, ADV DRUG RES, V13, P95
[7]  
MESNIL M, IN PRESS XENOBIOTICA
[8]  
MORELAND TA, 1986, DRUG METAB DISPOS, V14, P654
[9]   SELECTIVE INHIBITORY INTERACTIONS OF ALKOXYMETHYLENEDIOXYBENZENES TOWARDS MONO-OXYGENASE ACTIVITY IN RAT-HEPATIC MICROSOMES [J].
MURRAY, M ;
HETNARSKI, K ;
WILKINSON, CF .
XENOBIOTICA, 1985, 15 (05) :369-379
[10]  
POISSON M, 1984, ARZNEIMITTEL-FORSCH, V34-1, P199