2-ALKYL ANALOGS OF IDAZOXAN (RX-781094) WITH ENHANCED ANTAGONIST POTENCY AND SELECTIVITY AT CENTRAL ALPHA-2-ADRENOCEPTORS IN THE RAT

被引：17

作者：

GADIE, B

LANE, AC

MCCARTHY, PS

TULLOCH, IF

WALTER, DS

机构：

来源：

BRITISH JOURNAL OF PHARMACOLOGY | 1984年 / 83卷 / 03期

关键词：

D O I：

10.1111/j.1476-5381.1984.tb16224.x

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：707 / 712

页数：6

共 11 条

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[5] SELECTIVITY AND POTENCY OF 2-ALKYL ANALOGS OF THE ALPHA-2-ADRENOCEPTOR ANTAGONIST IDAZOXAN (RX-781094) IN PERIPHERAL SYSTEMS [J].

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[6] EVIDENCE FOR PHARMACOLOGICAL SIMILARITY BETWEEN ALPHA-2-ADRENOCEPTORS IN THE VAS-DEFERENS AND CENTRAL NERVOUS-SYSTEM OF THE RAT [J].

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BRITISH JOURNAL OF PHARMACOLOGY, 1983, 80 (01) :155-161

[7] STUDIES ON RX781094 - A SELECTIVE, POTENT AND SPECIFIC ANTAGONIST OF ALPHA-2-ADRENOCEPTORS [J].

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[8]

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[9]

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[10] THE EFFECTS OF METAL-IONS ON THE BINDING OF A NEW ALPHA-2-ADRENOCEPTOR ANTAGONIST RADIOLIGAND (H-3-RX-781094 IN RAT CEREBRAL-CORTEX [J].

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BIOCHEMICAL PHARMACOLOGY, 1983, 32 (20) :3122-3125

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