PRECLINICAL EVALUATION OF LOVASTATIN

被引:148
作者
MACDONALD, JS
GERSON, RJ
KORNBRUST, DJ
KLOSS, MW
PRAHALADA, S
BERRY, PH
ALBERTS, AW
BOKELMAN, DL
机构
[1] MERCK SHARP & DOHME RES LABS,DEPT BIOCHEM REGULAT,RAHWAY,NJ 07065
[2] CHIBRET,RIOM,FRANCE
关键词
D O I
10.1016/0002-9149(88)90003-3
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:J16 / J27
页数:12
相关论文
共 28 条
[1]   DISCOVERY, BIOCHEMISTRY AND BIOLOGY OF LOVASTATIN [J].
ALBERTS, AW .
AMERICAN JOURNAL OF CARDIOLOGY, 1988, 62 (15) :J10-J15
[2]   LACK OF CORRELATION BETWEEN RATE OF CHOLESTEROL-BIOSYNTHESIS AND ACTIVITY OF 3-HYDROXY-3-METHYLGLUTARYL COENZYME-A REDUCTASE IN RATS AND IN FIBROBLASTS TREATED WITH ML-236B [J].
BENSCH, WR ;
INGEBRITSEN, TS ;
DILLER, ER .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1978, 82 (01) :247-254
[3]  
BERRY PH, 1988, IN PRESS AM J PATHOL
[4]   BIOCHEMISTRY OF POLYISOPRENOID BIOSYNTHESIS [J].
BEYTIA, ED ;
PORTER, JW .
ANNUAL REVIEW OF BIOCHEMISTRY, 1976, 45 :113-142
[5]  
BROWN MS, 1980, J LIPID RES, V21, P505
[6]  
Clemmesen J., 1977, ACTA PATH MICROBIO S, V261, P38
[7]  
DRIVER HE, 1986, BRIT J EXP PATHOL, V67, P131
[8]  
DUGGAN DE, 1988, IN PRESS DRUG METAB
[9]  
ENDO A, 1979, BIOCHIM BIOPHYS ACTA, V575, P266
[10]   TESTICULAR FUNCTION IN TYPE-II HYPERLIPOPROTEINEMIC PATIENTS TREATED WITH LOVASTATIN (MEVINOLIN) OR NEOMYCIN [J].
FARNSWORTH, WH ;
HOEG, JM ;
MAHER, M ;
BRITTAIN, EH ;
SHERINS, RJ ;
BREWER, HB .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1987, 65 (03) :546-550