FORMATION OF INACTIVE CYTOCHROME-P-450 FE(II)-METABOLITE COMPLEXES WITH SEVERAL ERYTHROMYCIN DERIVATIVES BUT NOT WITH JOSAMYCIN AND MIDECAMYCIN IN RATS

被引:92
作者
LARREY, D [1 ]
TINEL, M [1 ]
PESSAYRE, D [1 ]
机构
[1] HOP BEAUJON,UNITE RECH PHYSIOPATHOL HEPAT,INSERM U24,F-92118 CLICHY,FRANCE
关键词
D O I
10.1016/0006-2952(83)90470-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1487 / 1493
页数:7
相关论文
共 27 条
[1]   POSSIBLE WARFARIN-ERYTHROMYCIN INTERACTION [J].
BARTLE, WR .
ARCHIVES OF INTERNAL MEDICINE, 1980, 140 (07) :985-987
[2]  
BRAZEAU P, 1970, PHARMACOL BASIS THER, P893
[3]  
BRAZIER JL, 1980, THERAPIE, V35, P545
[4]  
CUMMINS LH, 1977, PEDIATRICS, V59, P144
[5]  
DANAN G, 1981, J PHARMACOL EXP THER, V218, P509
[6]  
DRAVET C, 1977, LANCET, V1, P810
[7]   INHIBITION OF MIXED-FUNCTION OXIDATIONS BY SUBSTRATES FORMING REDUCED CYTOCHROME-P-450 METABOLIC-INTERMEDIATE COMPLEXES [J].
FRANKLIN, MR .
PHARMACOLOGY & THERAPEUTICS PART A-CHEMOTHERAPY TOXICOLOGY AND METABOLIC INHIBITORS, 1977, 2 (01) :227-245
[8]   COMPLEXES OF METABOLITES OF AMPHETAMINES WITH HEPATIC CYTOCHROME-P-450 [J].
FRANKLIN, MR .
XENOBIOTICA, 1974, 4 (03) :133-142
[9]  
GROLLEAU JY, 1981, THERAPIE, V36, P319
[10]  
Hayton A C, 1969, N Z Med J, V69, P42