A HIGH-AFFINITY, HIGHLY SELECTIVE LIGAND FOR THE DELTA OPIOID RECEPTOR - [H-3] [D-PEN2, PCL-PHE4, D-PEN5]ENKEPHALIN

被引：91

作者：

VAUGHN, LK

KNAPP, RJ

TOTH, G

WAN, YP

HRUBY, VJ

YAMAMURA, HI

机构：

[1] UNIV ARIZONA,DEPT PHARMACOL,TUCSON,AZ 85724

[2] UNIV ARIZONA,DEPT CHEM,TUCSON,AZ 85724

[3] NEW ENGLAND NUCL,BOSTON,MA 02118

来源：

LIFE SCIENCES | 1989年 / 45卷 / 11期

关键词：

D O I：

10.1016/0024-3205(89)90154-9

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

页码：1001 / 1008

页数：8

共 15 条

[1] CHARACTERIZATION OF [H-3][ 2-D-PENICILLAMINE, 5-D-PENICILLAMINE] ENKEPHALIN BINDING TO DELTA-OPIATE RECEPTORS IN THE RAT-BRAIN AND NEUROBLASTOMA-GLIOMA HYBRID CELL-LINE (NG-108-15) [J].

AKIYAMA, K ;

GEE, KW ;

MOSBERG, HI ;

HRUBY, VJ ;

YAMAMURA, HI .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (08) :2543-2547

[2]

[Anonymous], RECEPTORS

[3]

CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099

[4] THE USE OF [H-3]-[D-PEN2,D-PEN5]ENKEPHALIN AS A HIGHLY SELECTIVE LIGAND FOR THE DELTA-BINDING SITE [J].

COTTON, R ;

KOSTERLITZ, HW ;

PATERSON, SJ ;

RANCE, MJ ;

TRAYNOR, JR .

BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (04) :927-932

[5] COMPARATIVE BINDING-PROPERTIES OF LINEAR AND CYCLIC DELTA-SELECTIVE ENKEPHALIN ANALOGS - [H-3]-[D-THR2, LEU5] ENKEPHALYL-THR6 AND [H-3]-[D-PEN2, D-PEN5] ENKEPHALIN [J].

DELAYGOYET, P ;

ZAJAC, JM ;

RIGAUDY, P ;

FOUCAUD, B ;

ROQUES, BP .

FEBS LETTERS, 1985, 183 (02) :445-450

[6]

DELAYGOYET P, 1988, J BIOL CHEM, V263, P4124

[7]

HAWKINS KN, 1989, J PHARMACOL EXP THER, V248, P73

[8]

KRAMER T H, 1988, Society for Neuroscience Abstracts, V14, P33

[9]

LOWRY OH, 1951, J BIOL CHEM, V193, P265

[10]

LUI G K, 1988, Society for Neuroscience Abstracts, V14, P701

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