SYNTHESIS OF CYCLIC KETOMETHYLENE DIPEPTIDE DERIVATIVES

被引：8

作者：

DOMINGUEZ, MJ

GONZALEZMUNIZ, R

GARCIALOPEZ, MT

机构：

[1] Instituto de Química Médica, Juan de la Cierva

来源：

TETRAHEDRON | 1992年 / 48卷 / 13期

关键词：

D O I：

10.1016/S0040-4020(01)88534-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Methyl 6-aralkyl-2,5-diketopiperidine-3-carboxylates derived from L-Phe and L-Trp, and their 3-substituted analogues in which the 3-substituent is the side chain of Phe, Asp and Ala have been synthesized. Cycle[Trp-psi(COCH2)Gly] and cycle[Phe-psi(COCH2)-xi-Phe] have been also prepared.

引用

页码：2761 / 2772

页数：12

共 20 条

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