EQUILIBRIUM-ANALYSIS OF [H-3]TCP BINDING - EFFECTS OF GLYCINE, MAGNESIUM AND N-METHYL-D-ASPARTATE AGONISTS

被引:48
作者
JOHNSON, KM
SACAAN, AI
SNELL, LD
机构
关键词
D O I
10.1016/0014-2999(88)90845-X
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:141 / 146
页数:6
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[1]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[2]   PHENCYCLIDINE AND RELATED DRUGS BIND TO THE ACTIVATED N-METHYL-D-ASPARTATE RECEPTOR CHANNEL COMPLEX IN RAT-BRAIN MEMBRANES [J].
FAGG, GE .
NEUROSCIENCE LETTERS, 1987, 76 (02) :221-227
[3]   EXCITATORY AMINO-ACID SYNAPTIC MECHANISMS AND NEUROLOGICAL FUNCTION [J].
FAGG, GE ;
FOSTER, AC ;
GANONG, AH .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1986, 7 (09) :357-363
[4]   THE NOVEL ANTICONVULSANT MK-801 BINDS TO THE ACTIVATED STATE OF THE N-METHYL-D-ASPARTATE RECEPTOR IN RAT-BRAIN [J].
FOSTER, AC ;
WONG, EHF .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 91 (02) :403-409
[5]  
HARRISON NL, 1985, BR J PHARM, V84, P281
[6]   KETAMINE AND PHENCYCLIDINE CAUSE A VOLTAGE-DEPENDENT BLOCK OF RESPONSES TO L-ASPARTIC ACID [J].
HONEY, CR ;
MILJKOVIC, Z ;
MACDONALD, JF .
NEUROSCIENCE LETTERS, 1985, 61 (1-2) :135-139
[7]   QUANTITATIVE AUTORADIOGRAPHIC LOCALIZATION OF NMDA RECEPTORS IN RAT-BRAIN USING [H-3] CPP - COMPARISON WITH [H-3] TCP BINDING-SITES [J].
JARVIS, MF ;
MURPHY, DE ;
WILLIAMS, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 141 (01) :149-152
[8]   NONCOMPETITIVE REGULATION OF PHENCYCLIDINE SIGMA-RECEPTORS BY THE N-METHYL-D-ASPARTATE RECEPTOR ANTAGONIST D/(-)-2-AMINO-5-PHOSPHONOVALERIC ACID [J].
JAVITT, DC ;
JOTKOWITZ, A ;
SIRCAR, R ;
ZUKIN, SR .
NEUROSCIENCE LETTERS, 1987, 78 (02) :193-198
[9]   GLYCINE POTENTIATES THE NMDA RESPONSE IN CULTURED MOUSE-BRAIN NEURONS [J].
JOHNSON, JW ;
ASCHER, P .
NATURE, 1987, 325 (6104) :529-531
[10]  
JOHNSON KM, 1988, SIGMA PHENCYCLIDINE, P259