EVIDENCE OF A PEPTIDE BACKBONE CONTRIBUTION TOWARD SELECTIVE RECEPTOR RECOGNITION FOR LEUCINE ENKEPHALIN THIOAMIDE ANALOGS

被引：56

作者：

CLAUSEN, K

SPATOLA, AF

LEMIEUX, C

SCHILLER, PW

LAWESSON, SO

机构：

[1] CLIN RES INST MONTREAL, MONTREAL H2W 1R7, QUEBEC, CANADA

[2] AARHUS UNIV, DEPT ORGAN CHEM, DK-8000 AARHUS, DENMARK

来源：

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | 1984年 / 120卷 / 01期

关键词：

D O I：

10.1016/0006-291X(84)91449-9

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

收藏

页码：305 / 310

页数：6

相关论文

共 20 条

[1] CYCLIC AND ACYCLIC PARTIAL RETRO-INVERSO ENKEPHALINAMIDES - MU RECEPTOR SELECTIVE ENZYME RESISTANT ANALOGS
BERMAN, JM
GOODMAN, M
NGUYEN, TMD
SCHILLER, PW
[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 115 (03) : 864 - 870
[2] CLAUSEN K, 1984, J CHEM SOC P1
[3] CLAUSEN K, 1983, PEPTIDES 1982, P207
[4] SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION INVITRO OF CYCLIC ENKEPHALIN ANALOGS - EFFECT OF CONFORMATIONAL CONSTRAINTS ON OPIATE RECEPTOR SELECTIVITY
DIMAIO, J
NGUYEN, TMD
LEMIEUX, C
SCHILLER, PW
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (12) : 1432 - 1438
[5] A CYCLIC ENKEPHALIN ANALOG WITH HIGH INVITRO OPIATE ACTIVITY
DIMAIO, J
SCHILLER, PW
[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (12): : 7162 - 7166
[6] FOURNIEZALUSKI MC, 1981, MOL PHARM, V20, P481
[7] SYNTHESIS AND SOME PHARMACOLOGICAL PROPERTIES OF [1-DEAMINO,9-THIOGLYCINE]OXYTOCIN
JONES, WC
NESTOR, JJ
VIGNEAUD, VD
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1973, 95 (17) : 5677 - 5679
[8] LACOUR TFM, 1983, INT J PEPT PROT RES, V22, P509
[9] FACILE REGIOSELECTIVE FORMATION OF THIOPEPTIDE LINKAGES FROM OLIGOPEPTIDES WITH NEW THIONATION REAGENTS
LAJOIE, G
LEPINE, F
MAZIAK, L
BELLEAU, B
[J]. TETRAHEDRON LETTERS, 1983, 24 (36) : 3815 - 3818
[10] ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS
LORD, JAH
WATERFIELD, AA
HUGHES, J
KOSTERLITZ, HW
[J]. NATURE, 1977, 267 (5611) : 495 - 499