INVITRO BINDING-PROPERTIES AND AUTORADIOGRAPHIC IMAGING OF 3-IODOBENZAMIDE ([I-125] IBZM) - A POTENTIAL IMAGING LIGAND FOR D-2 DOPAMINE-RECEPTORS IN SPECT

被引:49
作者
BRUCKE, T [1 ]
TSAI, YF [1 ]
MCLELLAN, C [1 ]
SINGHANYOM, W [1 ]
KUNG, HF [1 ]
COHEN, RM [1 ]
CHIUEH, CC [1 ]
机构
[1] UNIV PENN,DEPT NUCL MED,PHILADELPHIA,PA 19104
关键词
D O I
10.1016/0024-3205(88)90123-3
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2097 / 2104
页数:8
相关论文
共 27 条
[1]   A DETAILED MAPPING OF DOPAMINE D-2 RECEPTORS IN RAT CENTRAL-NERVOUS-SYSTEM BY AUTORADIOGRAPHY WITH [I-125] IODOSULPRIDE [J].
BOUTHENET, ML ;
MARTRES, MP ;
SALES, N ;
SCHWARTZ, JC .
NEUROSCIENCE, 1987, 20 (01) :117-155
[2]  
BURT DR, 1976, MOL PHARMACOL, V12, P800
[3]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[4]  
CRAWLEY JCW, 1983, LANCET, V2, P975
[5]  
CRAWLEY JCW, 1986, LANCET, V2, P224
[6]  
DEPAULIS T, 1985, EUR J MED CHEM, V20, P273
[7]   SUBSTITUTED BENZAMIDES AS LIGANDS FOR VISUALIZATION OF DOPAMINE RECEPTOR-BINDING IN THE HUMAN-BRAIN BY POSITRON EMISSION TOMOGRAPHY [J].
FARDE, L ;
EHRIN, E ;
ERIKSSON, L ;
GREITZ, T ;
HALL, H ;
HEDSTROM, CG ;
LITTON, JE ;
SEDVALL, G .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (11) :3863-3867
[8]   QUANTITATIVE-ANALYSIS OF D2 DOPAMINE RECEPTOR-BINDING IN THE LIVING HUMAN-BRAIN BY PET [J].
FARDE, L ;
HALL, H ;
EHRIN, E ;
SEDVALL, G .
SCIENCE, 1986, 231 (4735) :258-261
[9]   SOME INVITRO RECEPTOR-BINDING PROPERTIES OF [H-3] ETICLOPRIDE, A NOVEL SUBSTITUTED BENZAMIDE, SELECTIVE FOR DOPAMINE-D2 RECEPTORS IN THE RAT-BRAIN [J].
HALL, H ;
KOHLER, C ;
GAWELL, L .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 111 (02) :191-199
[10]  
HAMON M, 1984, BRAIN RECEPTOR METHO, P309