SYNTHESIS OF PYRIMIDIN-2-ONE NUCLEOSIDES AS ACID-STABLE INHIBITORS OF CYTIDINE DEAMINASE

被引：68

作者：

KIM, CH

MARQUEZ, VE

MAO, DT

HAINES, DR

MCCORMACK, JJ

机构：

[1] NCI,DIV CANC TREATMENT,DEV THERAPEUT PROGRAM,PHARMACOL & EXPTL THERAPEUT LAB,BETHESDA,MD 20892

[2] UNIV VERMONT,COLL MED,DEPT PHARMACOL,BURLINGTON,VT 05401

[3] UNIV VERMONT,VERMONT REG CANC CTR,BURLINGTON,VT 05401

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 08期

关键词：

D O I：

10.1021/jm00158a009

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1374 / 1380

页数：7

共 33 条

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[9] SUBSTRATE-SPECIFICITY OF BACTERIAL THYMIDYLATE-SYNTHETASE
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[J]. COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS, 1974, 39 (06) : 1646 - 1661
[10] PREPARATION OF ANALOGS OF CYTOSINE AND 2-PYRIMIDINONE NUCLEOSIDES AND THEIR EFFECT ON BACTERIAL (ESCHERICHIA-COLI A19) CYTIDINE AMINOHYDROLASE
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[J]. COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS, 1985, 50 (02) : 393 - 417

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