EVIDENCE FOR AN INVOLVEMENT OF GABA RECEPTORS IN THE MEDIATION OF THE PROCONVULSANT ACTION OF ETHYL-BETA-CARBOLINE-3-CARBOXYLATE

被引:22
作者
CONCAS, A
SERRA, M
SALIS, M
NURCHI, V
CRISPONI, G
BIGGIO, G
机构
关键词
D O I
10.1016/0028-3908(84)90194-1
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:323 / 326
页数:4
相关论文
共 17 条
[1]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[2]   [H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS [J].
BRAESTRUP, C ;
NIELSEN, M .
JOURNAL OF NEUROCHEMISTRY, 1981, 37 (02) :333-341
[3]   BRAIN BENZODIAZEPINE RECEPTORS INCREASE AFTER CHRONIC ETHYL-BETA-CARBOLINE-3-CARBOXYLATE [J].
CONCAS, A ;
SALIS, M ;
BIGGIO, G .
LIFE SCIENCES, 1983, 32 (11) :1175-1182
[4]   ETHYL-BETA-CARBOLINE-3-CARBOXYLATE DECREASES [H-3]GABA BINDING IN MEMBRANE PREPARATIONS OF RAT CEREBRAL-CORTEX [J].
CONCAS, A ;
SALIS, M ;
SERRA, M ;
CORDA, MG ;
BIGGIO, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 89 (1-2) :179-181
[5]   BETA-CARBOLINES ENHANCE SHOCK-INDUCED SUPPRESSION OF DRINKING IN RATS [J].
CORDA, MG ;
BLAKER, WD ;
MENDELSON, WB ;
GUIDOTTI, A ;
COSTA, E .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (07) :2072-2076
[6]   MOLECULAR MECHANISMS IN THE RECEPTOR ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1979, 19 :531-545
[7]   ETHYL BETA-CARBOLINE CARBOXYLATE LOWERS SEIZURE THRESHOLD AND ANTAGONIZES FLURAZEPAM-INDUCED SEDATION IN RATS [J].
COWEN, PJ ;
GREEN, AR ;
NUTT, DJ ;
MARTIN, IL .
NATURE, 1981, 290 (5801) :54-55
[8]   GAMMA-AMINOBUTYRIC ACID REGULATION OF THE BENZODIAZEPINE RECEPTOR - BIOCHEMICAL-EVIDENCE FOR PHARMACOLOGICALLY DIFFERENT EFFECTS OF BENZODIAZEPINES AND PROPYL BETA-CARBOLINE-3-CARBOXYLATE [J].
EHLERT, FJ ;
ROESKE, WR ;
BRAESTRUP, C ;
YAMAMURA, SH ;
YAMAMURA, HI .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (04) :593-595
[9]  
HIRSCH S, 1982, PHARM BIOCH BEHAV, V16, P245
[10]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265