STEREOSELECTIVE BLOCKADE AT THE 5-HT AUTORECEPTOR AND INHIBITION OF RADIOLIGAND BINDING TO CENTRAL 5-HT RECOGNITION SITES BY THE OPTICAL ISOMERS OF METHIOTHEPIN

被引：35

作者：

HIBERT, M

MIDDLEMISS, DN

机构：

[1] CONTINENTAL PHARMA,PARC SCI LOUVAIN LA NEUVE,RUE GRANDBONPRE 2,B-1348 MT ST GUIBERT,BELGIUM

[2] MERRELL DOW RES INST,STRASBOURG CTR,F-67084 STRASBOURG,FRANCE

来源：

NEUROPHARMACOLOGY | 1986年 / 25卷 / 01期

关键词：

D O I：

10.1016/0028-3908(86)90050-X

中图分类号：

Q189 [神经科学];

学科分类号：

071006 ;

摘要：

引用

页码：1 / 4

页数：4

共 17 条

[1] SEROTONIN RELEASE IS MODULATED BY PRESYNAPTIC AUTORECEPTORS [J].

CERRITO, F ;

RAITERI, M .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 57 (04) :427-430

[2] PRESYNAPTIC REGULATION OF NEUROTRANSMITTER RELEASE IN THE BRAIN - FACTS AND HYPOTHESIS [J].

CHESSELET, MF .

NEUROSCIENCE, 1984, 12 (02) :347-375

[3] CHARACTERIZATION OF 5-HYDROXYTRYPTAMINERGIC AUTORECEPTORS IN THE RAT HYPOTHALAMUS [J].

COX, B ;

ENNIS, C .

JOURNAL OF PHARMACY AND PHARMACOLOGY, 1982, 34 (07) :438-441

[4] EVIDENCE FOR COMMON PHARMACOLOGICAL PROPERTIES OF [H-3]5-HYDROXYTRYPTAMINE BINDING-SITES, PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE AUTORECEPTORS IN CNS AND INHIBITORY PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE RECEPTORS ON SYMPATHETIC-NERVES [J].

ENGEL, G ;

GOTHERT, M ;

MULLERSCHWEINITZER, E ;

SCHLICKER, E ;

SISTONEN, L ;

STADLER, PA .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 324 (02) :116-124

[5] A CUMULATIVE DOSE-RESPONSE TECHNIQUE FOR THE CHARACTERIZATION OF PRE-SYNAPTIC RECEPTORS MODULATING [3H]NORADRENALIN RELEASE FROM RAT-BRAIN SLICES [J].

FRANKHUYZEN, AL ;

MULDER, AH .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 78 (01) :91-97

[6] EXTRACELLULAR 5-HYDROXYTRYPTAMINE INHIBITS 5-HYDROXYTRYPTAMINE RELEASE FROM RAT-BRAIN CORTEX SLICES [J].

GOTHERT, M ;

WEINHEIMER, G .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 310 (01) :93-96

[7] AUTORECEPTOR-MEDIATED INHIBITION OF H-3-5-HYDROXYTRYPTAMINE RELEASE FROM RAT-BRAIN CORTEX SLICES BY ANALOGS OF 5-HYDROXYTRYPTAMINE [J].

GOTHERT, M ;

SCHLICKER, E .

LIFE SCIENCES, 1983, 32 (11) :1183-1191

[8]

JACQUES J, 1971, TETRAHEDRON LETT, V48, P4617

[9] PRESYNAPTIC RECEPTORS AND MODULATION OF NEUROTRANSMISSION - PHARMACOLOGICAL IMPLICATIONS AND THERAPEUTIC RELEVANCE [J].

LANGER, SZ .

TRENDS IN NEUROSCIENCES, 1980, 3 (05) :110-112

[10] RECEPTOR-BINDING PROFILE OF R-41-468, A NOVEL ANTAGONIST AT 5-HT2 RECEPTORS [J].

LEYSEN, JE ;

AWOUTERS, F ;

KENNIS, L ;

LADURON, PM ;

VANDENBERK, J ;

JANSSEN, PAJ .

LIFE SCIENCES, 1981, 28 (09) :1015-1022

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