DESACETYL-1-NANTRADOL - A SELECTIVE PROSTAGLANDIN ANTAGONIST

被引:8
作者
HORNE, WC
机构
[1] BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
[2] HARVARD UNIV,SCH MED,BOSTON,MA 02115
来源
PROSTAGLANDINS LEUKOTRIENES AND MEDICINE | 1984年 / 15卷 / 01期
关键词
D O I
10.1016/0262-1746(84)90063-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:129 / 136
页数:8
相关论文
共 22 条
[1]   CHARACTERIZATION OF HUMAN PLATELET ALPHA-ADRENERGIC RECEPTOR - CORRELATION OF [H-3] DIHYDROERGOCRYPTINE BINDING WITH AGGREGATION AND ADENYLATE-CYCLASE INHIBITION [J].
ALEXANDER, RW ;
COOPER, B ;
HANDIN, RI .
JOURNAL OF CLINICAL INVESTIGATION, 1978, 61 (05) :1136-1144
[2]   ON THE MULTIPLICITY OF PLATELET PROSTAGLANDIN RECEPTORS .1. EVALUATION OF COMPETITIVE ANTAGONISM BY AGGREGOMETRY [J].
ANDERSEN, NH ;
EGGERMAN, TL ;
HARKER, LA ;
WILSON, CH ;
DE, B .
PROSTAGLANDINS, 1980, 19 (05) :711-735
[3]   MOLECULAR-BASIS FOR PROSTAGLANDIN POTENCY .3. TESTS OF THE SIGNIFICANCE OF THE HAIRPIN CONFORMATION IN BIORECOGNITION PHENOMENA [J].
ANDERSEN, NH ;
IMAMOTO, S ;
SUBRAMANIAN, N ;
PICKER, DH ;
LADNER, DW ;
DE, B ;
TYNAN, SS ;
EGGERMAN, TL ;
HARKER, LA ;
ROBERTSON, RP ;
OIEN, HG ;
RAO, CV .
PROSTAGLANDINS, 1981, 22 (05) :841-856
[4]  
Bennett A, 1974, Adv Drug Res, V8, P83
[5]   MORPHINE-LIKE DRUGS INHIBIT STIMULATION BY E PROSTAGLANDINS OF CYCLIC-AMP FORMATION BY RAT-BRAIN HOMOGENATE [J].
COLLIER, HOJ ;
ROY, AC .
NATURE, 1974, 248 (5443) :24-27
[6]   SYNTHESIS AND CHIROPTICAL CHARACTERIZATION OF PROSTACYCLIN DIASTEREOMERS [J].
DE, B ;
ANDERSEN, NH ;
IPPOLITO, RM ;
WILSON, CH ;
JOHNSON, WD .
PROSTAGLANDINS, 1980, 19 (02) :221-247
[7]  
DeTitta G T, 1980, Adv Prostaglandin Thromboxane Res, V6, P381
[8]   EVALUATION OF INTRAMUSCULAR LEVONANTRADOL AND PLACEBO IN ACUTE POSTOPERATIVE PAIN [J].
JAIN, AK ;
RYAN, JR ;
MCMAHON, FG ;
SMITH, G .
JOURNAL OF CLINICAL PHARMACOLOGY, 1981, 21 (8-9) :S320-S326
[9]   STRUCTURE ACTIVITY STUDIES LEADING TO A TISSUE-SELECTIVE HYPOTENSIVE PROSTAGLANDIN ANALOG, 13,14-DIHYDRO-16-PHENYL-OMEGA-TETRANOR PGE2 [J].
JOHNSON, MR ;
SCHAAF, TK ;
CONSTANTINE, JW ;
HESS, HJ .
PROSTAGLANDINS, 1980, 20 (03) :515-520
[10]   STUDIES ON THE CHARACTERIZATION OF PROSTANOID RECEPTORS - A PROPOSED CLASSIFICATION [J].
KENNEDY, I ;
COLEMAN, RA ;
HUMPHREY, PPA ;
LEVY, GP ;
LUMLEY, P .
PROSTAGLANDINS, 1982, 24 (05) :667-689