MARKED AND PROLONGED INHIBITION OF MAMMALIAN ORNITHINE DECARBOXYLASE INVIVO BY ESTERS OF (E)-2-(FLUOROMETHYL)DEHYDROORNITHINE

被引：24

作者：

MAMONT, PS ^{[1
]}

DANZIN, C ^{[1
]}

KOLB, M ^{[1
]}

GERHART, F ^{[1
]}

BEY, P ^{[1
]}

SJOERDSMA, A ^{[1
]}

机构：

[1] MERRELL DOW RES INST,CINCINNATI,OH 45215

来源：

BIOCHEMICAL PHARMACOLOGY | 1986年 / 35卷 / 02期

关键词：

D O I：

10.1016/0006-2952(86)90509-5

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：159 / 165

页数：7

共 26 条

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[2] BARTHOLEYNS J, 1984, CANCER RES, V44, P4972
[3] ALPHA-(FLUOROMETHYL)DEHYDROORNITHINE AND ALPHA-(FLUOROMETHYL)DEHYDROPUTRESCINE ANALOGS AS IRREVERSIBLE INHIBITORS OF ORNITHINE DECARBOXYLASE
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[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1983, 26 (11) : 1551 - 1556
[4] CATALYTIC IRREVERSIBLE INHIBITION OF TRYPANOSOMA-BRUCEI-BRUCEI ORNITHINE DECARBOXYLASE BY SUBSTRATE AND PRODUCT ANALOGS AND THEIR EFFECTS ON MURINE TRYPANOSOMIASIS
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[J]. BIOCHEMICAL PHARMACOLOGY, 1985, 34 (10) : 1773 - 1777
[5] (2R,5R)-6-HEPTYNE-2,5-DIAMINE, AN EXTREMELY POTENT INHIBITOR OF MAMMALIAN ORNITHINE DECARBOXYLASE
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[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 116 (01) : 237 - 243
[6] EFFECT ON PROSTATIC GROWTH OF 2-DIFLUOROMETHYLORNITHINE, AN EFFECTIVE INHIBITOR OF ORNITHINE DECARBOXYLASE
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CLAVERIE, N
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[J]. BIOCHEMICAL JOURNAL, 1982, 202 (01) : 175 - 181
[7] EFFECT OF ALPHA-DIFLUOROMETHYLORNITHINE, AN ENZYME-ACTIVATED IRREVERSIBLE INHIBITOR OF ORNITHINE DECARBOXYLASE, ON POLYAMINE LEVELS IN RAT TISSUES
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BEY, P
[J]. LIFE SCIENCES, 1979, 24 (06) : 519 - 524
[8] FOZARD JR, 1980, SCIENCE, V208, P505
[9] INHIBITORY-ACTION OF ALPHA-DIFLUOROMETHYLORNITHINE ON RODENT MALARIA (PLASMODIUM-BERGHEI)
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HERMAN, F
[J]. TRANSACTIONS OF THE ROYAL SOCIETY OF TROPICAL MEDICINE AND HYGIENE, 1982, 76 (06) : 776 - 777
[10] ASSAY OF ALPHA-DIFLUOROMETHYLORNITHINE IN BODY-FLUIDS AND TISSUES BY AUTOMATIC AMINO-ACID-ANALYSIS
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[J]. JOURNAL OF CHROMATOGRAPHY, 1981, 223 (02): : 409 - 416

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