VINYLOGOUS CARBINOLAMINE TUMOR INHIBITORS .21. SYNTHESIS, CHEMICAL-REACTIVITY, AND ANTILEUKEMIC ACTIVITY OF 5-SUBSTITUTED 6,7-BIS(HYDROXYMETHYL)PYRROLO[1,2-C]THIAZOLE BISCARBAMATES AND THE CORRESPONDING SULFOXIDES AND SULFONES

被引：32

作者：

ANDERSON, WK

MACH, RH

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 11期

关键词：

D O I：

10.1021/jm00394a030

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2109 / 2115

页数：7

共 9 条

[1]

ANDERSON WK, 1982, CANCER TREAT REP, V66, P91

[2]

ANDERSON WK, 1980, ARZNEIMITTEL-FORSCH, V30-1, P765

[3] SELECTIVE REDUCTION OF CARBOXYLIC-ACID ESTERS IN THE PRESENCE OF A 5-MEMBERED CYCLIC SULFONE [J].

ANDERSON, WK ;

MACH, RH .

SYNTHETIC COMMUNICATIONS, 1986, 16 (08) :911-915

[4]

ANDERSON WK, 1982, CANCER RES, V42, P2168

[5] VINYLOGOUS CARBINOLAMINE TUMOR INHIBITORS .20. COMPARISON OF THE CHEMICAL REACTIVITIES AND ANTINEOPLASTIC ACTIVITIES OF ALPHA,BETA, ALPHA,BETA', BETA,BETA', AND ALPHA,ALPHA'-BIS[[[(2-PROPYLAMINO)CARBONYL]OXY]METHYL]-SUBSTITUTED PYRROLES [J].

ANDERSON, WK ;

HEIDER, AR .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (11) :2392-2395

[6] SYNTHESIS AND ANTILEUKEMIC ACTIVITY OF 5-SUBSTITUTED 2,3-DIHYDRO-6,7-BIS(HYDROXYMETHYL)-1H-PYRROLIZINE DIESTERS [J].

ANDERSON, WK ;

COREY, PF .

JOURNAL OF MEDICINAL CHEMISTRY, 1977, 20 (06) :812-818

[7] A STUDY OF COMPARATIVE CHEMICAL AND BIOLOGICAL ACTIVITIES OF ALKYLATING AGENTS [J].

BARDOS, TJ ;

DATTAGUP.N ;

HEBBORN, P ;

TRIGGLE, DJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1965, 8 (02) :167-&

[8]

Hansch C, 1979, SUBSTITUENT CONSTANT

[9] STEREOSPECIFIC SYNTHESIS OF 1-SUBSTITUTED PYRROLIZIDINES [J].

PIZZORNO, MT ;

ALBONICO, SM .

JOURNAL OF ORGANIC CHEMISTRY, 1974, 39 (05) :731-731

← 1 →