PILOCARPIC ACID-ESTERS AS NOVEL SEQUENTIALLY LABILE PILOCARPINE PRODRUGS FOR IMPROVED OCULAR DELIVERY

被引：36

作者：

BUNDGAARD, H

FALCH, E

LARSEN, C

MOSHER, GL

MIKKELSON, TJ

机构：

[1] ROYAL DANISH SCH PHARM,DEPT PHARMACEUT,DK-2100 COPENHAGEN,DENMARK

[2] UNIV KANSAS,SCH PHARM,DEPT PHARMACEUT CHEM,LAWRENCE,KS 66045

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 08期

关键词：

D O I：

10.1021/jm00146a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：979 / 981

页数：3

共 17 条

[1] ANDERSON JA, 1980, INVEST OPHTH VIS SCI, V19, P817
[2] OCULAR PENETRATION OF PILOCARPINE IN PRIMATES
ASSEFF, CF
WEISMAN, RL
PODOS, SM
BECKER, B
[J]. AMERICAN JOURNAL OF OPHTHALMOLOGY, 1973, 75 (02) : 212 - 215
[3] VISUAL EFFECTS OF PILOCARPINE IN GLAUCOMA - COMPARATIVE-STUDY OF ADMINISTRATION BY EYEDROPS OR BY OCULAR THERAPEUTIC SYSTEMS
BROWN, HS
MELTZER, G
MERRILL, RC
FISHER, M
FERRE, C
PLACE, VA
[J]. ARCHIVES OF OPHTHALMOLOGY, 1976, 94 (10) : 1716 - 1719
[4] HYDROLYSIS AND EPIMERIZATION KINETICS OF PILOCARPINE IN BASIC AQUEOUS-SOLUTION AS DETERMINED BY HPLC
BUNDGAARD, H
HANSEN, SH
[J]. INTERNATIONAL JOURNAL OF PHARMACEUTICS, 1982, 10 (04) : 281 - 289
[5] PRO-DRUGS AS DRUG DELIVERY SYSTEMS .17. ESTERS OF 4-HYDROXYBUTYRIC ACIDS AS POTENTIAL PRO-DRUG TYPES FOR GAMMA-LACTONES
BUNDGAARD, H
LARSEN, C
[J]. INTERNATIONAL JOURNAL OF PHARMACEUTICS, 1980, 7 (02) : 169 - 176
[6] CORNEAL PERMEATION OF TOPICAL PILOCARPINE NITRATE IN RABBIT
CHRAI, SS
ROBINSON, JR
[J]. AMERICAN JOURNAL OF OPHTHALMOLOGY, 1974, 77 (05) : 735 - 739
[7] LACRIMAL AND INSTILLED FLUID DYNAMICS IN RABBIT EYES
CHRAI, SS
PATTON, TF
MEHTA, A
ROBINSON, JR
[J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1973, 62 (07) : 1112 - 1121
[8] PRODRUG APPROACHES TO ENHANCEMENT OF PHYSICOCHEMICAL PROPERTIES OF DRUGS .4. NOVEL EPINEPHRINE PRODRUG
HUSSAIN, A
TRUELOVE, JE
[J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1976, 65 (10) : 1510 - 1512
[9] MECHANISTIC AND QUANTITATIVE-EVALUATION OF PRE-CORNEAL PILOCARPINE DISPOSITION IN ALBINO RABBITS
LEE, VHL
ROBINSON, JR
[J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1979, 68 (06) : 673 - 684
[10] OPHTHALMIC SOLUTION BUFFER SYSTEMS .1. THE EFFECT OF BUFFER CONCENTRATION ON THE OCULAR ABSORPTION OF PILOCARPINE
MITRA, AK
MIKKELSON, TJ
[J]. INTERNATIONAL JOURNAL OF PHARMACEUTICS, 1982, 10 (03) : 219 - 229

← 1 2 →