EFFECT OF OMEGA-CONOTOXIN GVIA ON CA-2+ INFLUX AND ENDOGENOUS ACETYLCHOLINE-RELEASE FROM CHICKEN BRAIN PREPARATIONS

被引:22
作者
LUNDY, PM [1 ]
STAUDERMAN, K [1 ]
GOULET, JC [1 ]
FREW, R [1 ]
机构
[1] MERRELL DOW PHARMACEUT INC,RES INST,DIV BIOCHEM SCI,CINCINNATI,OH 45215
关键词
D O I
10.1016/0197-0186(89)90008-9
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:49 / 54
页数:6
相关论文
共 21 条
[1]   EFFECTS OF POTASSIUM, VERATRIDINE AND SCORPION-VENOM ON CALCIUM ACCUMULATION AND TRANSMITTER RELEASE BY NERVE-TERMINALS INVITRO [J].
BLAUSTEIN, MP .
JOURNAL OF PHYSIOLOGY-LONDON, 1975, 247 (03) :617-655
[2]   DIHYDROPYRIDINE CALCIUM-CHANNEL ANTAGONIST BINDING IN NONMAMMALIAN VERTEBRATES - CHARACTERIZATION AND RELATIONSHIP TO PERIPHERAL-TYPE BINDING-SITES FOR BENZODIAZEPINES [J].
BOLGER, GT ;
WEISSMAN, BA ;
LUEDDENS, H ;
BARRETT, JE ;
WITKIN, J ;
PAUL, SM ;
SKOLNICK, P .
BRAIN RESEARCH, 1986, 368 (02) :351-356
[3]  
BRADFORD MM, 1976, ANAL BIOCHEM, V116, P48
[4]   CENTRAL INTERACTIONS BETWEEN DIHYDROPYRIDINES AND CHOLINERGIC SYSTEMS IN THE CONTROL OF BLOOD-PRESSURE IN RAT [J].
BRISAC, AM ;
HUGUET, F ;
CHAMPEROUX, P ;
MONTASTRUC, JL ;
LUCET, B ;
GERARD, P ;
LAURENT, S ;
NARCISSE, G ;
SCHMITT, H .
BRAIN RESEARCH, 1987, 435 (1-2) :160-166
[5]  
CRUZ LJ, 1986, J BIOL CHEM, V261, P6230
[6]   FAILURE OF THE CALCIUM-CHANNEL ACTIVATOR, BAY K-8644, TO INCREASE THE RELEASE OF ACETYLCHOLINE FROM NERVE-TERMINALS IN BRAIN AND DIAPHRAGM [J].
DOLEZAL, V ;
TUCEK, S .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 91 (03) :475-479
[7]   INHIBITION OF CENTRAL NEUROTRANSMITTER RELEASE BY OMEGA-CONOTOXIN GVIA, A PEPTIDE MODULATOR OF THE N-TYPE VOLTAGE-SENSITIVE CALCIUM-CHANNEL [J].
DOOLEY, DJ ;
LUPP, A ;
HERTTING, G .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1987, 336 (04) :467-470
[8]   STEREOSELECTIVITY AT THE CALCIUM-CHANNEL - OPPOSITE ACTION OF THE ENANTIOMERS OF A 1,4-DIHYDROPYRIDINE [J].
HOF, RP ;
RUEGG, UT ;
HOF, A ;
VOGEL, A .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1985, 7 (04) :689-693
[9]   APPLICATION TO MAMMALIAN-TISSUES OF THE CHEMI-LUMINESCENT METHOD FOR DETECTING ACETYLCHOLINE [J].
ISRAEL, M ;
LESBATS, B .
JOURNAL OF NEUROCHEMISTRY, 1982, 39 (01) :248-250
[10]   1,4-DIHYDROPYRIDINE CA-2+ CHANNEL ANTAGONISTS AND ACTIVATORS - A COMPARISON OF BINDING CHARACTERISTICS WITH PHARMACOLOGY [J].
JANIS, RA ;
TRIGGLE, DJ .
DRUG DEVELOPMENT RESEARCH, 1984, 4 (03) :257-274