MIXING-TANK MODEL FOR PREDICTING DISSOLUTION RATE CONTROL OF ORAL ABSORPTION

被引:115
作者
DRESSMAN, JB
FLEISHER, D
机构
关键词
D O I
10.1002/jps.2600750202
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:109 / 116
页数:8
相关论文
共 29 条
[1]   BIOAVAILABILITY AND RELATED HEART FUNCTION INDEX OF DIGOXIN CAPSULES AND TABLETS IN CARDIAC PATIENTS [J].
ASTORRI, E ;
BIANCHI, G ;
LACANNA, G ;
ASSANELLI, D ;
VISIOLI, O ;
MARZO, A .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1979, 68 (01) :104-106
[2]  
ATKINSON R. M., 1962, ANTIBIOT AND CHEMOTHER, V12, P232
[3]   ABSORPTION CHARACTERISTICS OF SOLID DISPERSED AND MICRONIZED GRISEOFULVIN IN MAN [J].
CHIOU, WL ;
RIEGELMAN, S .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1971, 60 (09) :1376-+
[5]  
DILLARD RL, 1965, GASTROENTEROLOGY, V49, P58
[6]   ABSORPTION POTENTIAL - ESTIMATING THE FRACTION ABSORBED FOR ORALLY-ADMINISTERED COMPOUNDS [J].
DRESSMAN, JB ;
AMIDON, GL ;
FLEISHER, D .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1985, 74 (05) :588-589
[7]   PHYSICOCHEMICAL MODEL FOR DOSE-DEPENDENT DRUG ABSORPTION [J].
DRESSMAN, JB ;
FLEISHER, D ;
AMIDON, GL .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1984, 73 (09) :1274-1279
[8]  
DRESSMAN JB, UNPUB DIG DIS SCI
[9]   CHANGES IN CRYSTALLINITY AND SOLUBILITY ON COMMINUTION OF DIGOXIN AND OBSERVATIONS ON SPIRONOLACTONE AND ESTRADIOL [J].
FLORENCE, AT ;
SALOLE, EG .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1976, 28 (08) :637-642
[10]   A MATHEMATICAL-MODEL OF DRUG ABSORPTION [J].
GOODACRE, BC ;
MURRAY, PJ .
JOURNAL OF CLINICAL AND HOSPITAL PHARMACY, 1981, 6 (02) :117-133