INHIBITION OF THE UTEROTROPIC ACTIVITY OF ESTROGENS AND ANTI-ESTROGENS BY THE SHORT-ACTING ANTIESTROGEN-LY117018

被引:60
作者
JORDAN, VC
GOSDEN, B
机构
关键词
D O I
10.1210/endo-113-2-463
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
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页码:463 / 468
页数:6
相关论文
共 18 条
[1]   MOLECULAR BASIS FOR DRUG ACTION [J].
ARIENS, EJ ;
SIMONIS, AM .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1964, 16 (03) :137-&
[2]   UTERINE BIOASSAY OF TAMOXIFEN, TRIOXIFENE AND A NEW ESTROGEN ANTAGONIST (LY117018) IN RATS AND MICE [J].
BLACK, LJ ;
GOODE, RL .
LIFE SCIENCES, 1980, 26 (17) :1453-1458
[3]   EVIDENCE FOR BIOLOGICAL ACTION OF THE ANTI-ESTROGENS LY117018 AND TAMOXIFEN BY DIFFERENT MECHANISMS [J].
BLACK, LJ ;
GOODE, RL .
ENDOCRINOLOGY, 1981, 109 (03) :987-989
[4]   ANTI-ESTROGEN SPECIFIC, HIGH-AFFINITY SATURABLE BINDING-SITES IN RAT UTERINE CYTOSOL [J].
FAYE, JC ;
LASSERRE, B ;
BAYARD, F .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 93 (04) :1225-1231
[5]  
GREENBLATT RB, 1952, AM J OBSTET GYNECOL, V63, P1361
[6]   BINDING OF [H-3] MONOHYDROXYTAMOXIFEN BY IMMATURE RAT-TISSUES INVIVO [J].
JORDAN, VC ;
BOWSERFINN, RA .
ENDOCRINOLOGY, 1982, 110 (04) :1281-1291
[7]   DOSE-RELATED EFFECTS OF NON-STEROIDAL ANTIOESTROGENS AND ESTROGENS ON MEASUREMENT OF CYTOPLASMIC ESTROGEN RECEPTORS IN RAT AND MOUSE UTERUS [J].
JORDAN, VC ;
ROWSBY, L ;
DIX, CJ ;
PRESTWICH, G .
JOURNAL OF ENDOCRINOLOGY, 1978, 78 (01) :71-81
[8]   MONOHYDROXYLATED METABOLITE OF TAMOXIFEN WITH POTENT ANTI-ESTROGENIC ACTIVITY [J].
JORDAN, VC ;
COLLINS, MM ;
ROWSBY, L ;
PRESTWICH, G .
JOURNAL OF ENDOCRINOLOGY, 1977, 75 (02) :305-316
[9]   EVALUATION OF THE ANTI-TUMOR ACTIVITY OF THE NON-STEROIDAL ANTIOESTROGEN MONOHYDROXYTAMOXIFEN IN THE DMBA-INDUCED RAT MAMMARY-CARCINOMA MODEL [J].
JORDAN, VC ;
ALLEN, KE .
EUROPEAN JOURNAL OF CANCER, 1980, 16 (02) :239-251
[10]   NON-STEROIDAL ANTI-ESTROGENS - THEIR BIOLOGICAL EFFECTS AND POTENTIAL MECHANISMS OF ACTION [J].
JORDAN, VC ;
DIX, CJ ;
NAYLOR, KE ;
PRESTWICH, G ;
ROWSBY, L .
JOURNAL OF TOXICOLOGY AND ENVIRONMENTAL HEALTH, 1978, 4 (2-3) :363-390