EVIDENCE FOR DIFFERENT STATES OF THE DOPAMINE D1 RECEPTOR - CLOZAPINE AND FLUPERLAPINE MAY PREFERENTIALLY LABEL AN ADENYLATE CYCLASE-COUPLED STATE OF THE D1-RECEPTOR

被引:105
作者
ANDERSEN, PH [1 ]
BRAESTRUP, C [1 ]
机构
[1] ST HANS MENTAL HOSP, PSYCHOPHARMACOL RES LAB, DK-4000 ROSKILDE, DENMARK
关键词
D O I
10.1111/j.1471-4159.1986.tb13094.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1822 / 1831
页数:10
相关论文
共 29 条
[1]   EFFECT OF CLOZAPINE ON TURNOVER OF DOPAMINE IN CORPUS STRIATUM AND IN LIMBIC SYSTEM [J].
ANDEN, N ;
STOCK, G .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1973, 25 (04) :346-348
[2]   A COMPARISON BETWEEN DOPAMINE-STIMULATED ADENYLATE-CYCLASE AND H-3-SCH-23390 BINDING IN RAT STRIATUM [J].
ANDERSEN, PH ;
GRONVALD, FC ;
JANSEN, JA .
LIFE SCIENCES, 1985, 37 (21) :1971-1983
[3]   SPECIFIC BINDING OF H-3 SCH 23390 TO DOPAMINE D1 RECEPTORS INVIVO [J].
ANDERSEN, PH ;
GRONVALD, FC .
LIFE SCIENCES, 1986, 38 (16) :1507-1514
[4]   SOME ATYPICAL NEUROLEPTICS INHIBIT [H-3] SCH 23390 BINDING INVIVO [J].
ANDERSEN, PH ;
NIELSEN, EB ;
GRONVALD, FC ;
BRAESTRUP, C .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 120 (01) :143-144
[6]  
BARNETT A, 1986, Drugs of the Future, V11, P49
[7]   CHARACTERIZATION OF THE BINDING OF H-3-SCH 23390, A SELECTIVE D-1 RECEPTOR ANTAGONIST LIGAND, IN RAT STRIATUM [J].
BILLARD, W ;
RUPERTO, V ;
CROSBY, G ;
IORIO, LC ;
BARNETT, A .
LIFE SCIENCES, 1984, 35 (18) :1885-1893
[8]  
BROWN JH, 1984, J BIOL CHEM, V259, P3777
[9]   DOPAMINE-SENSITIVE ADENYLATE CYCLASE IN MAMMALIAN BRAIN - POSSIBLE SITE OF ACTION OF ANTIPSYCHOTIC-DRUGS [J].
CLEMENTC.YC ;
KEBABIAN, JW ;
PETZOLD, GL ;
GREENGARD, P .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1974, 71 (04) :1113-1117
[10]   NEUROLEPTIC ACTION OF CLOZAPINE INJECTED INTO VARIOUS BRAIN AREAS IN RATS [J].
FOG, R .
INTERNATIONAL PHARMACOPSYCHIATRY, 1975, 10 (02) :89-93