SOLUBILIZATION OF BRAIN BENZODIAZEPINE RECEPTORS WITH A ZWITTERIONIC DETERGENT - OPTIMAL PRESERVATION OF THEIR FUNCTIONAL INTERACTION WITH THE GABA RECEPTORS

被引:41
作者
MERNOFF, ST [1 ]
CHERWINSKI, HM [1 ]
BECKER, JW [1 ]
DEBLAS, AL [1 ]
机构
[1] SUNY STONY BROOK,DEPT NEUROBIOL & BEHAV,STONY BROOK,NY 11794
关键词
D O I
10.1111/j.1471-4159.1983.tb04804.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:752 / 758
页数:7
相关论文
共 32 条
[1]   SOLUBLE GAMMA-AMINOBUTYRIC ACID AND BENZODIAZEPINE RECEPTORS FROM RAT CEREBRAL-CORTEX [J].
ASANO, T ;
OGASAWARA, N .
LIFE SCIENCES, 1981, 29 (02) :193-200
[2]   SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].
BRAESTRUP, C ;
SQUIRES, RF .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809
[3]   INFLUENCE OF GABA RECEPTOR AGONISTS AND ANTAGONISTS ON BINDING OF DIAZEPAM-H-3 TO BENZODIAZEPINE RECEPTOR [J].
BRILEY, MS ;
LANGER, SZ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 52 (01) :129-132
[4]  
BURCH TP, 1981, P NATL ACAD SCI-BIOL, V78, P3945, DOI 10.1073/pnas.78.6.3945
[5]   MOLECULAR MECHANISMS IN THE RECEPTOR ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1979, 19 :531-545
[6]   IS THE BENZODIAZEPINE RECEPTOR COUPLED TO A CHLORIDE ANION CHANNEL [J].
COSTA, T ;
RODBARD, D ;
PERT, CB .
NATURE, 1979, 277 (5694) :315-317
[7]   EFFECT OF GABAERGIC DRUGS ON BENZODIAZEPINE BINDING-SITE SENSITIVITY IN RAT CEREBRAL-CORTEX [J].
GALLAGER, DW ;
THOMAS, JW ;
TALLMAN, JF .
BIOCHEMICAL PHARMACOLOGY, 1978, 27 (23) :2745-2749
[8]   SOLUBILIZATION OF HISTAMINE H-1, GABA AND BENZODIAZEPINE RECEPTORS [J].
GAVISH, M ;
CHANG, RSL ;
SNYDER, SH .
LIFE SCIENCES, 1979, 25 (09) :783-789
[9]   GAMMA-AMINOBUTYRIC ACID AND BENZODIAZEPINE RECEPTORS - COPURIFICATION AND CHARACTERIZATION [J].
GAVISH, M ;
SNYDER, SH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (03) :1939-1942
[10]   SOLUBLE BENZODIAZEPINE RECEPTORS - GABAERGIC REGULATION [J].
GAVISH, M ;
SNYDER, SH .
LIFE SCIENCES, 1980, 26 (08) :579-582