A POTENT NONPEPTIDE CHOLECYSTOKININ ANTAGONIST SELECTIVE FOR PERIPHERAL-TISSUES ISOLATED FROM ASPERGILLUS-ALLIACEUS

被引：320

作者：

CHANG, RSL

LOTTI, VJ

MONAGHAN, RL

BIRNBAUM, J

STAPLEY, EO

GOETZ, MA

ALBERSSCHONBERG, G

PATCHETT, AA

LIESCH, JM

HENSENS, OD

SPRINGER, JP

机构：

[1] MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065

[2] MERCK SHARP & DOHME RES LABS,DEPT NEW LEAD DISCOVERY,RAHWAY,NJ 07065

[3] MERCK SHARP & DOHME RES LABS,DEPT ANALYT NAT PROD CHEM,RAHWAY,NJ 07065

[4] MERCK SHARP & DOHME RES LABS,DEPT BIOPHYS,RAHWAY,NJ 07065

来源：

SCIENCE | 1985年 / 230卷 / 4722期

关键词：

D O I：

10.1126/science.2994227

中图分类号：

O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];

学科分类号：

07 ; 0710 ; 09 ;

摘要：

引用

页码：177 / 179

页数：3

共 20 条

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[4] FURTHER EVIDENCE THAT SUBSTANCE-P PARTLY MEDIATES THE ACTION OF CHOLECYSTOKININ OCTAPEPTIDE (CCK-8) ON THE GUINEA-PIG ILEUM BUT NOT GALLBLADDER - STUDIES WITH A SUBSTANCE-P ANTAGONIST
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[J]. NEUROSCIENCE LETTERS, 1984, 46 (01) : 71 - 75
[5] INACTIVATION OF CHOLECYSTOKININ RECEPTORS IN RAT PANCREATIC MEMBRANES BY SULFHYDRYL-REAGENTS - PROTECTION BY GUANOSINE 5'-TRIPHOSPHATE (GTP) BUT NOT N-2, O-2-DIBUTYRYL GUANOSINE 3',5'-CYCLIC-MONOPHOSPHATE (DIBUTYRYL CGMP)
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[J]. BIOCHEMICAL PHARMACOLOGY, 1984, 33 (14) : 2334 - 2335
[6] COMPARISON OF INVIVO AND INVITRO RESPONSES TO SULFATED AND NON-SULFATED CERULETIDE
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[J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 47 (03) : 359 - 363
[7] CHOLECYSTOKININ RECEPTOR ANTAGONISTS
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[J]. AMERICAN JOURNAL OF PHYSIOLOGY, 1984, 246 (05): : G471 - G476
[8] GOETZ MA, UNPUB
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[10] DISTINCT CHOLECYSTOKININ RECEPTORS IN BRAIN AND PANCREAS
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[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (11): : 6917 - 6921

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