METHOCTRAMINE, A POLYMETHYLENE TETRAAMINE, DIFFERENTIATES 3 SUBTYPES OF MUSCARINIC RECEPTOR IN DIRECT BINDING-STUDIES

被引:105
作者
MICHEL, AD
WHITING, RL
机构
关键词
D O I
10.1016/0014-2999(88)90349-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:61 / 66
页数:6
相关论文
共 16 条
[1]  
BURGEN ASV, 1984, TIPS S, V5, P1
[2]  
CASSINELLI A, 1987, 1986 P INT S CHOL MU
[3]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[4]   [H-3]-LABELED RAUWOLSCINE AND [H-3]-LABELED YOHIMBINE BINDING TO RAT CEREBRAL AND HUMAN-PLATELET MEMBRANES - POSSIBLE HETEROGENEITY OF ALPHA-2-ADRENOCEPTORS [J].
CHEUNG, YD ;
BARNETT, DB ;
NAHORSKI, SR .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 84 (1-2) :79-85
[5]   ACTION OF AGONISTS AND ANTAGONISTS AT MUSCARINIC RECEPTORS PRESENT ON ILEUM AND ATRIA INVITRO [J].
CLAGUE, RU ;
EGLEN, RM ;
STRACHAN, AC ;
WHITING, RL .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 86 (01) :163-170
[6]  
DEJONGE A, 1986, BRIT J PHARMACOL, V89, pP551
[7]   MUSCARINIC RECEPTOR SUBTYPES - M1 AND M2 BIOCHEMICAL AND FUNCTIONAL-CHARACTERIZATION [J].
HAMMER, R ;
GIACHETTI, A .
LIFE SCIENCES, 1982, 31 (26) :2991-2998
[8]   BINDING PROFILE OF A NOVEL CARDIOSELECTIVE MUSCARINE RECEPTOR ANTAGONIST, AF-DX 116, TO MEMBRANES OF PERIPHERAL-TISSUES AND BRAIN IN THE RAT [J].
HAMMER, R ;
GIRALDO, E ;
SCHIAVI, GB ;
MONFERINI, E ;
LADINSKY, H .
LIFE SCIENCES, 1986, 38 (18) :1653-1662
[9]   PIRENZEPINE DISTINGUISHES BETWEEN DIFFERENT SUBCLASSES OF MUSCARINIC RECEPTORS [J].
HAMMER, R ;
BERRIE, CP ;
BIRDSALL, NJM ;
BURGEN, ASV ;
HULME, EC .
NATURE, 1980, 283 (5742) :90-92
[10]   DIFFERENTIAL BLOCKADE OF MUSCARINIC RECEPTOR SUBTYPES BY POLYMETHYLENE TETRAAMINES - NOVEL CLASS OF SELECTIVE ANTAGONISTS OF CARDIAC M-2 MUSCARINIC RECEPTORS [J].
MELCHIORRE, C ;
CASSINELLI, A ;
QUAGLIA, W .
JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (01) :201-204