MAGNESIUM REDUCES AFFINITIES OF ANTAGONISTS AT RAT CORTEX ALPHA-2-ADRENERGIC RECEPTORS LABELED WITH H-3-LABELED CLONIDINE - EVIDENCE FOR HETEROGENEITY OF ALPHA-2-RECEPTOR CONFORMATIONS WITH RESPECT TO ANTAGONISTS

被引:40
作者
SALAMA, AI [1 ]
LIN, LL [1 ]
REPP, LD [1 ]
UPRICHARD, DC [1 ]
机构
[1] NORTHWESTERN UNIV,DEPT PHARMACOL,CHICAGO,IL 60611
关键词
D O I
10.1016/0024-3205(82)90693-2
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:1305 / 1311
页数:7
相关论文
共 19 条
[1]  
COLQUHOUN D, 1973, DRUG RECEPTORS, P149, DOI DOI 10.1007/978-1-349-00910-7_11
[2]   HUMAN-PLATELET ALPHA-2-ADRENERGIC RECEPTORS - LABELING WITH YOHIMBINE-H-3, A SELECTIVE ANTAGONIST LIGAND [J].
DAIGUJI, M ;
MELTZER, HY ;
UPRICHARD, DC .
LIFE SCIENCES, 1981, 28 (24) :2705-2717
[3]  
DELEAN A, MOL PHARM NEUROTRANS
[4]   REGULATION OF MUSCARINIC RECEPTOR-BINDING BY GUANINE-NUCLEOTIDES AND N-ETHYLMALEIMIDE [J].
EHLERT, FJ ;
ROESKE, WR ;
YAMAMURA, HI .
JOURNAL OF SUPRAMOLECULAR STRUCTURE, 1980, 14 (02) :149-162
[5]   ROLE OF PHOSPHATIDYLINOSITOL TURNOVER IN ALPHA1 AND OF ADENYLATE-CYCLASE INHIBITION IN ALPHA2 EFFECTS OF CATECHOLAMINES [J].
FAIN, JN ;
GARCIASAINZ, JA .
LIFE SCIENCES, 1980, 26 (15) :1183-1194
[6]   ALPHA-2-ADRENOCEPTORS IN RAT-BRAIN - THE DIVALENT-CATION SITE [J].
GLOSSMANN, H ;
HORNUNG, R .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 314 (02) :101-109
[7]   RADIOLIGAND BINDING-STUDIES OF ADRENERGIC-RECEPTORS - NEW INSIGHTS INTO MOLECULAR AND PHYSIOLOGICAL REGULATION [J].
HOFFMAN, BB ;
LEFKOWITZ, RJ .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1980, 20 :581-608
[8]   AGONIST VERSUS ANTAGONIST BINDING TO ALPHA-ADRENERGIC RECEPTORS [J].
HOFFMAN, BB ;
MICHEL, T ;
KILPATRICK, DM ;
LEFKOWITZ, RJ ;
TOLBERT, MEM ;
GILMAN, H ;
FAIN, JN .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (08) :4569-4573
[9]  
HOFFMAN BB, 1980, J BIOL CHEM, V255, P4645
[10]  
KAHN D, 1982, MOL PHARM