CALCIUM-CHANNEL RECEPTOR-BINDING STUDIES FOR DILTIAZEM AND ITS MAJOR METABOLITES - FUNCTIONAL CORRELATION TO INHIBITION OF PORTAL-VEIN MYOGENIC ACTIVITY

被引:48
作者
SCHOEMAKER, H [1 ]
HICKS, PE [1 ]
LANGER, SZ [1 ]
机构
[1] LABS ETUDES & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
关键词
D O I
10.1097/00005344-198702000-00008
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:173 / 180
页数:8
相关论文
共 35 条
[1]   SPECIFIC BINDING OF [H-3] D-CIS-DILTIAZEM TO CARDIAC SARCOLEMMA AND ITS INHIBITION BY CALCIUM [J].
BALWIERCZAK, JL ;
SCHWARTZ, A .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 116 (1-2) :193-194
[2]  
BOLES RG, 1984, J PHARMACOL EXP THER, V229, P333
[3]  
BOLGER GT, 1983, J PHARMACOL EXP THER, V225, P291
[4]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[5]   SPECIFIC BINDING OF [H-3]LABELED NITRENDIPINE TO MEMBRANES FROM CORONARY-ARTERIES AND HEART IN RELATION TO PHARMACOLOGICAL EFFECTS - PARADOXICAL STIMULATION BY DILTIAZEM [J].
DEPOVER, A ;
MATLIB, MA ;
LEE, SW ;
DUBE, GP ;
GRUPP, IL ;
GRUPP, G ;
SCHWARTZ, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 108 (01) :110-117
[6]   THE BINDING OF [H-3]-LABELED NITRENDIPINE TO RECEPTORS FOR CALCIUM-CHANNEL ANTAGONISTS IN THE HEART, CEREBRAL-CORTEX, AND ILEUM OF RATS [J].
EHLERT, FJ ;
ROESKE, WR ;
ITOGA, E ;
YAMAMURA, HI .
LIFE SCIENCES, 1982, 30 (25) :2191-2202
[7]   [H-3] VERAPAMIL BINDING-SITES IN SKELETAL-MUSCLE TRANSVERSE TUBULE MEMBRANES [J].
GALIZZI, JP ;
FOSSET, M ;
LAZDUNSKI, M .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 118 (01) :239-245
[8]   MOLECULAR PHARMACOLOGY OF THE CALCIUM-CHANNEL - EVIDENCE FOR SUBTYPES, MULTIPLE DRUG-RECEPTOR SITES, CHANNEL SUBUNITS, AND THE DEVELOPMENT OF A RADIOIODINATED 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL LABEL, [I-125] IODIPINE [J].
GLOSSMANN, H ;
FERRY, DR ;
GOLL, A ;
ROMBUSCH, M .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1984, 6 :S608-S621
[9]   TEMPERATURE-DEPENDENT REGULATION OF D-CIS-[H-3] DILTIAZEM BINDING TO CA-2+ CHANNELS BY 1,4-DIHYDROPYRIDINE CHANNEL AGONISTS AND ANTAGONISTS [J].
GLOSSMANN, H ;
LINN, T ;
ROMBUSCH, M ;
FERRY, DR .
FEBS LETTERS, 1983, 160 (1-2) :226-232
[10]  
GOLENHOFEN K, 1970, PFLUGERS ARCH, V34, P312