NEW CARBOXYALKYL INHIBITORS OF BRAIN ENKEPHALINASE - SYNTHESIS, BIOLOGICAL-ACTIVITY, AND ANALGESIC PROPERTIES

被引：41

作者：

FOURNIEZALUSKI, MC

CHAILLET, P

SOROCALUCAS, E

MARCAISCOLLADO, H

COSTENTIN, J

ROQUES, BP

机构：

[1] CNRS, DEPT CHIM ORGAN, ERA 613, F-75270 PARIS 06, FRANCE

[2] INSERM, SC 21, UER SCI PHARMACEUT & BIOL, F-75006 PARIS, FRANCE

[3] UNIV ROUEN, UER MED & PHARM, PHARMACODYNAM LAB, F-76800 ST ETIENNE DU ROU, FRANCE

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1983年 / 26卷 / 01期

关键词：

D O I：

10.1021/jm00355a013

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：60 / 65

页数：6

共 43 条

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[9] DESIGN OF POTENT COMPETITIVE INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYME - CARBOXYALKANOYL AND MERCAPTOALKANOYL AMINO-ACIDS
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[J]. BIOCHEMISTRY, 1977, 16 (25) : 5484 - 5491
[10] CHEMISTRY AND PHARMACOLOGY OF THE METHADOLS AND ACETYLMETHADOLS
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