AN EXAMINATION OF THE OPIATE RECEPTOR SUBTYPES LABELED BY [H-3]CYCLOFOXY - AN OPIATE ANTAGONIST SUITABLE FOR POSITRON EMISSION TOMOGRAPHY

被引:29
作者
ROTHMAN, RB
MCLEAN, S
机构
[1] NIMH, PRECLIN PHARMACOL LAB, BETHESDA, MD USA
[2] NIMH, NEUROPHYSIOL LAB, BETHESDA, MD USA
[3] ST ELIZABETHS HOSP, WASHINGTON, DC 20032 USA
关键词
D O I
10.1016/0006-3223(88)90016-9
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:435 / 458
页数:24
相关论文
共 55 条
[1]  
ACETO MD, 1985, NIDA RES MONOGR, V67, P442
[2]   INTERCONVERTING MU-FORMS AND DELTA-FORMS OF THE OPIATE RECEPTOR IN RAT STRIATAL PATCHES [J].
BOWEN, WD ;
GENTLEMAN, S ;
HERKENHAM, M ;
PERT, CB .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (08) :4818-4822
[3]  
BURKE TR, 1985, HETEROCYCLES, V23, P99
[4]  
CASCIERI MA, 1985, J BIOL CHEM, V260, P1501
[5]  
CHENEY BV, 1982, MOL PHARMACOL, V22, P349
[6]   DYNORPHIN1-8 AND DYNORPHIN1-9 ARE LIGANDS FOR THE KAPPA-SUBTYPE OF OPIATE RECEPTOR [J].
CORBETT, AD ;
PATERSON, SJ ;
MCKNIGHT, AT ;
MAGNAN, J ;
KOSTERLITZ, HW .
NATURE, 1982, 299 (5878) :79-81
[7]  
CREESE I, 1975, J PHARMACOL EXP THER, V194, P205
[8]   A COMPARATIVE AUTORADIOGRAPHIC STUDY OF THE DISTRIBUTIONS OF SUBSTANCE-P AND ELEDOISIN BINDING-SITES IN RAT-BRAIN [J].
DANKS, JA ;
ROTHMAN, RB ;
CASCIERI, MA ;
CHICCHI, GG ;
LIANG, T ;
HERKENHAM, M .
BRAIN RESEARCH, 1986, 385 (02) :273-281
[9]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[10]  
FROST JJ, 1985, J COMPUT ASSIST TOMO, V9, P231, DOI 10.1097/00004728-198503000-00001