IRREVERSIBLE BLOCKADE OF CENTRAL 5-HT BINDING-SITES BY 8-METHOXY-2'-CHLORO-PAT

被引:23
作者
EMERIT, MB [1 ]
GOZLAN, H [1 ]
HALL, MD [1 ]
HAMON, M [1 ]
MARQUET, A [1 ]
机构
[1] COLL FRANCE,CHAIRE NEUROPHARMACOL,INSERM,U114,F-75231 PARIS 05,FRANCE
关键词
D O I
10.1016/0006-2952(85)90770-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:883 / 892
页数:10
相关论文
共 36 条
  • [1] SYNTHESIS OF ALKOXY-1,2,3,4-TETRAHYDRONAPHTHALENE DERIVATIVES .I. 2-AMINO-, ALKYLAMINO-, AND DIALKYLAMINO-DERIVATIVES
    AMES, DE
    EVANS, D
    GREY, TF
    ISLIP, PJ
    RICHARDS, KE
    [J]. JOURNAL OF THE CHEMICAL SOCIETY, 1965, (APR): : 2636 - &
  • [2] 8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN, A NEW CENTRALLY ACTING 5-HYDROXYTRYPTAMINE RECEPTOR AGONIST
    ARVIDSSON, LE
    HACKSELL, U
    NILSSON, JLG
    HJORTH, S
    CARLSSON, A
    LINDBERG, P
    SANCHEZ, D
    WIKSTROM, H
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (08) : 921 - 923
  • [3] BENNETT JP, 1976, MOL PHARMACOL, V12, P373
  • [4] PHOTOAFFINITY-LABELING OF SEROTONIN-BINDING PROTEINS
    CHENG, SH
    SHIH, JC
    [J]. LIFE SCIENCES, 1979, 25 (26) : 2197 - 2203
  • [5] APORPHINES .50. KINETICS OF SOLVOLYSIS OF N-(2-CHLOROETHYL)NORAPOMORPHINE, AN IRREVERSIBLE DOPAMINE RECEPTOR ANTAGONIST
    COHEN, SA
    NEUMEYER, JL
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1983, 26 (10) : 1348 - 1353
  • [6] CORTES R, 1984, British Journal of Pharmacology, V82, p202P
  • [7] DERMER O, 1969, ETHYLENIMINE OTHER A
  • [8] ALTERATIONS IN CENTRAL NEUROTRANSMITTER RECEPTOR-BINDING SITES FOLLOWING ESTRADIOL IMPLANTATION IN FEMALE RATS
    GOETZ, C
    BOURGOIN, S
    CESSELIN, F
    BRANDI, A
    BRESSION, D
    MARTINET, M
    PEILLON, F
    HAMON, M
    [J]. NEUROCHEMISTRY INTERNATIONAL, 1983, 5 (04) : 375 - 383
  • [9] IDENTIFICATION OF PRE-SYNAPTIC SEROTONIN AUTORECEPTORS USING A NEW LIGAND - H-3-PAT
    GOZLAN, H
    ELMESTIKAWY, S
    PICHAT, L
    GLOWINSKI, J
    HAMON, M
    [J]. NATURE, 1983, 305 (5930) : 140 - 142
  • [10] TURNOVER OF SPECIFIC [H-3]SPIPERONE AND [H-3]N,NORMAL-PROPYLNORAPOMORPHINE BINDING-SITES IN RAT STRIATUM FOLLOWING PHENOXYBENZAMINE ADMINISTRATION
    HALL, MD
    JENNER, P
    MARSDEN, CD
    [J]. BIOCHEMICAL PHARMACOLOGY, 1983, 32 (19) : 2973 - 2977