6-CHLORO-2,3,4,5-TETRAHYDRO-3-METHYL-1H-3-BENZAZEPINE - A POTENT AND SELECTIVE ANTAGONIST OF ALPHA-2-ADRENOCEPTORS

被引：24

作者：

DEMARINIS, RM ^{[1
]}

HIEBLE, JP ^{[1
]}

MATTHEWS, WD ^{[1
]}

机构：

[1] SK&F LABS,DEPT PHARMACOL,PHILADELPHIA,PA 19101

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1983年 / 26卷 / 09期

关键词：

D O I：

10.1021/jm00363a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1213 / 1214

页数：2

共 10 条

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SMITH, CFC ;

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[3]

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[5] PRESYNAPTIC RECEPTORS AND MODULATION OF NEUROTRANSMISSION - PHARMACOLOGICAL IMPLICATIONS AND THERAPEUTIC RELEVANCE [J].

LANGER, SZ .

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[6]

STARKE K, 1977, REV PHYSL BIOCH PHAR, V71, P1

[7]

STARKE K, ADV BIOSCI, V18, P1

[8] ALPHA-2 ADRENOCEPTORS - CLASSIFICATION, LOCALIZATION, MECHANISMS, AND TARGETS FOR DRUGS [J].

TIMMERMANS, PBMWM ;

VANZWIETEN, PA .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (12) :1389-1401

[9]

Wikberg J E, 1979, Acta Physiol Scand Suppl, V468, P1

[10]

1974, Patent No. 3804849

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