SYNTHESIS AND REACTIVITY OF 2-(1,3-DITHIAN-2-YL)INDOLES .4. INFLUENCE OF THE N,N-DIETHYLCARBAMOYL INDOLE PROTECTING GROUP

被引：12

作者：

CASTELLS, J ^{[1
]}

TROIN, Y ^{[1
]}

DIEZ, A ^{[1
]}

RUBIRALTA, M ^{[1
]}

GRIERSON, DS ^{[1
]}

HUSSON, HP ^{[1
]}

机构：

[1] CNRS,INST CHIM SUBSTANCES NAT,F-91198 GIF SUR YVETTE,FRANCE

来源：

TETRAHEDRON | 1991年 / 47卷 / 37期

关键词：

2-(1,3-DITHIAN-2-YL)INDOLES; INDOLE; N; N-DIETHYLCARBAMOYL PROTECTING GROUP;

D O I：

10.1016/S0040-4020(01)81946-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The effect of the N,N-diethylcarbamoyl indole protecting group on the reactivity of 2-(1,3-dithian-2-yl)indole 7 in front of a series of electrophiles, as well as the potential synthetic usefulness of the resulting 2,2-disubstituted dithianes is reported.

引用

页码：7911 / 7924

页数：14

共 18 条

[1] BENNASAR ML, 1990, TETRAHEDRON LETT, V31, P1893
[2] BENNASAR ML, 1989, HETEROCYCLES, V29, P745
[3] COMINS DL, 1986, TETRAHEDRON LETT, V27, P1869, DOI 10.1016/S0040-4039(00)84397-X
[4] NEW METHODS FOR ALKALOID SYNTHESIS - GENERATION OF INDOLE-2, 3-DIQUINOMETHANES AS A ROUTE TO INDOLE ALKALOIDS
GALLAGHER, T
MAGNUS, P
[J]. TETRAHEDRON, 1981, 37 (23) : 3889 - 3897
[5] GENERATION AND RING-OPENING OF 2,3-DILITHIO-1-(PHENYLSULFONYL)INDOLE
GRIBBLE, GW
SAULNIER, MG
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1983, 48 (04) : 607 - 609
[6] HO TL, 1985, TETRAHEDRON, V41, P1
[7] JOHNSON DA, 1986, HETEROCYCLES, V24, P2127
[8] INDOLE-2,3-QUINODIMETHANES - SYNTHESIS OF SELECTIVELY PROTECTED DERIVATIVES OF THE FUSED DIMERIC INDOLE ALKALOID STAUROSPORINONE
MAGNUS, PD
SEAR, NL
[J]. TETRAHEDRON, 1984, 40 (14) : 2795 - 2797
[9] SYNTHESIS AND REACTIVITY OF 2-(1',3'-DITHIAN-2'-YL)INDOLES
RUBIRALTA, M
CASAMITJANA, N
GRIERSON, DS
HUSSON, HP
[J]. TETRAHEDRON, 1988, 44 (02) : 443 - 450
[10] SYNTHETIC APPLICATIONS OF 2-(1,3-DITHIAN-2-YL)INDOLES - A NEW SYNTHETIC APPROACH TO STRYCHNOS ALKALOIDS
RUBIRALTA, M
TORRENS, A
REIG, I
GRIERSON, DS
HUSSON, HP
[J]. HETEROCYCLES, 1989, 29 (11) : 2121 - 2133

← 1 2 →