TACHYKININ RECEPTOR ANTAGONISTS AND POTENTIAL CLINICAL-APPLICATIONS AT PERIPHERAL LEVEL

被引:16
作者
MAGGI, CA
PATACCHINI, R
ROVERO, P
GIULIANI, S
GIACHETTI, A
机构
关键词
D O I
10.1042/bst0190909
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:909 / 912
页数:4
相关论文
共 27 条
  • [1] SEARCH FOR A PHYSIOLOGICAL-ROLE OF SUBSTANCE-P IN GASTROINTESTINAL MOTILITY
    BARTHO, L
    HOLZER, P
    [J]. NEUROSCIENCE, 1985, 16 (01) : 1 - 32
  • [2] [LEU9-PSI(CH2NH)LEU10]-NEUROKININ-A(4-10) (MDL-28,564) DISTINGUISHES TISSUE TACHYKININ PEPTIDE NK2 RECEPTORS
    BUCK, SH
    HARBESON, SL
    HASSMANN, CF
    SHATZER, SA
    ROUISSI, N
    NANTEL, F
    VANGIERSBERGEN, PLM
    [J]. LIFE SCIENCES, 1990, 47 (10) : PL37 - PL41
  • [3] STRUCTURE-ACTIVITY STUDY OF NEUROKININS - ANTAGONISTS FOR THE NEUROKININ-2 RECEPTOR
    DION, S
    ROUISSI, N
    NANTEL, F
    JUKIC, D
    RHALEB, NE
    TOUSIGNANT, C
    TELEMAQUE, S
    DRAPEAU, G
    REGOLI, D
    NALINE, E
    ADVENIER, C
    ROVERO, P
    MAGGI, CA
    [J]. PHARMACOLOGY, 1990, 41 (04) : 184 - 194
  • [4] BIOLOGICAL EVALUATION OF SUBSTANCE-P ANTAGONISTS
    FOLKERS, K
    HAKANSON, R
    HORIG, J
    CHENG, XJ
    LEANDER, S
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (02) : 449 - 456
  • [5] SPECIES-DIFFERENCES IN AFFINITIES OF NONPEPTIDE ANTAGONISTS FOR SUBSTANCE-P RECEPTORS
    GITTER, BD
    WATERS, DC
    BRUNS, RF
    MASON, NR
    NIXON, JA
    HOWBERT, JJ
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1991, 197 (2-3) : 237 - 238
  • [6] IDENTIFICATION OF NEUROTRANSMITTERS REGULATING INTESTINAL PERISTALTIC REFLEX IN HUMANS
    GRIDER, JR
    [J]. GASTROENTEROLOGY, 1989, 97 (06) : 1414 - 1419
  • [7] TACHYKININ RECEPTOR TYPES - CLASSIFICATION AND MEMBRANE SIGNALING MECHANISMS
    GUARD, S
    WATSON, SP
    [J]. NEUROCHEMISTRY INTERNATIONAL, 1991, 18 (02) : 149 - 165
  • [8] HAGAN RM, 1990, BRIT J PHARMACOL, V99, pP62
  • [10] MULTIPLE TACHYKININ BINDING-SITES IN PERIPHERAL-TISSUES AND IN BRAIN
    LEE, CM
    CAMPBELL, NJ
    WILLIAMS, BJ
    IVERSEN, LL
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 130 (03) : 209 - 217