SYNTHESIS AND RADIORECEPTOR BINDING-ACTIVITY OF N-0437, A NEW, EXTREMELY POTENT AND SELECTIVE D2 DOPAMINE RECEPTOR AGONIST

被引：66

作者：

HORN, AS ^{[1
]}

TEPPER, P ^{[1
]}

VANDERWEIDE, J ^{[1
]}

WATANABE, M ^{[1
]}

GRIGORIADIS, D ^{[1
]}

SEEMAN, P ^{[1
]}

机构：

[1] UNIV TORONTO,DEPT PHARMACOL,TORONTO M5S 1A8,ONTARIO,CANADA

来源：

PHARMACEUTISCH WEEKBLAD-SCIENTIFIC EDITION | 1985年 / 7卷 / 05期

关键词：

D O I：

10.1007/BF02307578

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：208 / 211

页数：4

共 18 条

[1] SYNTHESIS OF ALKOXY-1,2,3,4-TETRAHYDRONAPHTHALENE DERIVATIVES .I. 2-AMINO-, ALKYLAMINO-, AND DIALKYLAMINO-DERIVATIVES
AMES, DE
EVANS, D
GREY, TF
ISLIP, PJ
RICHARDS, KE
[J]. JOURNAL OF THE CHEMICAL SOCIETY, 1965, (APR): : 2636 - &
[2] N,N-DISUBSTITUTED 2-AMINOTETRALINS ARE POTENT D-2 DOPAMINE RECEPTOR AGONISTS
BEAULIEU, M
ITOH, Y
TEPPER, P
HORN, AS
KEBABIAN, JW
[J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 105 (1-2) : 15 - 21
[3] A COMPARISON OF THE POTENCIES OF VARIOUS DOPAMINE RECEPTOR AGONISTS IN MODELS FOR PRE-SYNAPTIC AND POSTSYNAPTIC RECEPTOR ACTIVITY
FEENSTRA, MGP
SUMNERS, C
GOEDEMOED, JH
DEVRIES, JB
ROLLEMA, H
HORN, AS
[J]. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 324 (02) : 108 - 115
[4] THE DOPAMINE NEUROLEPTIC RECEPTOR
GRIGORIADIS, D
SEEMAN, P
[J]. CANADIAN JOURNAL OF NEUROLOGICAL SCIENCES, 1984, 11 (01) : 108 - 113
[5] N-ALKYLATED 2-AMINOTETRALINS - CENTRAL DOPAMINE-RECEPTOR STIMULATING ACTIVITY
HACKSELL, U
SVENSSON, U
NILSSON, JLG
HJORTH, S
CARLSSON, A
WIKSTROM, H
LINDBERG, P
SANCHEZ, D
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1979, 22 (12) : 1469 - 1475
[6] N-0434, A VERY POTENT AND SPECIFIC NEW D-2 DOPAMINE RECEPTOR AGONIST
HORN, AS
TEPPER, P
KEBABIAN, JW
BEART, PM
[J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 99 (01) : 125 - 126
[7] HORN AS, 1984, Patent No. 4465692
[8] JANSSEN PAJ, 1968, DRUGS AFFECTING CENT, P37
[9] MULTIPLE RECEPTORS FOR DOPAMINE
KEBABIAN, JW
CALNE, DB
[J]. NATURE, 1979, 277 (5692) : 93 - 96
[10] LIGAND - A VERSATILE COMPUTERIZED APPROACH FOR CHARACTERIZATION OF LIGAND-BINDING SYSTEMS
MUNSON, PJ
RODBARD, D
[J]. ANALYTICAL BIOCHEMISTRY, 1980, 107 (01) : 220 - 239

← 1 2 →