THE ABSORPTION OF BETA-ADRENOCEPTOR ANTAGONISTS IN RAT INSITU SMALL-INTESTINE - THE EFFECT OF LIPOPHILICITY

被引:65
作者
TAYLOR, DC
POWNALL, R
BURKE, W
机构
关键词
D O I
10.1111/j.2042-7158.1985.tb05064.x
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:280 / 283
页数:4
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共 13 条
[1]  
COLLINS RF, 1976, BRIT J CLIN PHARMACO, V3, pP346
[2]   THE CLINICAL IMPORTANCE OF CARDIOSELECTIVITY AND LIPOPHILICITY IN BETA-BLOCKERS [J].
CRUICKSHANK, JM .
AMERICAN HEART JOURNAL, 1980, 100 (02) :160-178
[3]   DRUG ABSORPTION .I. AN IN SITU RAT GUT TECHNIQUE YIELDING REALISTIC ABSORPTION RATES [J].
DOLUISIO, JT ;
BILLUPS, NF ;
DITTERT, LW ;
SUGITA, ET ;
SWINTOSKY, JV .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1969, 58 (10) :1196-+
[4]   METABOLIC STUDIES IN PATIENTS WITH NADOLOL - ORAL AND INTRAVENOUS ADMINISTRATION [J].
DREYFUSS, J ;
BRANNICK, LJ ;
VUKOVICH, RA ;
SHAW, JM ;
WILLARD, DA .
JOURNAL OF CLINICAL PHARMACOLOGY, 1977, 17 (5-6) :300-307
[5]  
FOURTILLAN JB, 1981, THERAPIE, V38, P457
[6]   ELIMINATION OF DRUGS BY ACTIVE INTESTINAL TRANSPORT [J].
GEORGE, CF ;
GRUCHY, BS .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1979, 31 (09) :643-644
[7]  
HIGUCHI WI, 1979, DRUG ABSORPTION, V21, P35
[8]  
Ho N.F.H., 1983, ANIMAL MODELS ORAL D, P27
[9]   DETERMINATION OF ACID SURFACE PH INVIVO IN RAT PROXIMAL JEJUNUM [J].
LUCAS, M .
GUT, 1983, 24 (08) :734-739
[10]  
MCAINSH J, 1977, POSTGRAD MED J, V53, P74