SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF NEW ARYLFLUORONAPHTHYRIDINE ANTIBACTERIAL AGENTS

被引：84

作者：

CHU, DTW

FERNANDES, PB

CLAIBORNE, AK

GRACEY, EH

PERNET, AG

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 11期

关键词：

D O I：

10.1021/jm00161a036

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2363 / 2369

页数：7

共 14 条

[1]

Albrecht R, 1977, Prog Drug Res, V21, P9

[2] SYNTHESIS AND STRUCTURE ACTIVITY RELATIONSHIPS OF NOVEL ARYLFLUOROQUINOLONE ANTIBACTERIAL AGENTS [J].

CHU, DTW ;

FERNANDES, PB ;

CLAIBORNE, AK ;

PIHULEAC, E ;

NORDEEN, CW ;

MALECZKA, RE ;

PERNET, AG .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (11) :1558-1564

[3] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF BENZOTHIAZOLO[3,2-A]QUINOLONE ANTIBACTERIAL AGENTS [J].

CHU, DTW ;

FERNANDES, PB ;

PERNET, AG .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (08) :1531-1534

[4]

GOUEFFON Y, 1981, CR ACAD SCI III-VIE, V292, P37

[5] TRIMMED SPEARMAN-KARBER METHOD FOR ESTIMATING MEDIAN LETHAL CONCENTRATIONS IN TOXICITY BIOASSAYS [J].

HAMILTON, MA ;

RUSSO, RC ;

THURSTON, RV .

ENVIRONMENTAL SCIENCE & TECHNOLOGY, 1977, 11 (07) :714-719

[6] STRUCTURE-ACTIVITY-RELATIONSHIPS OF ANTI-BACTERIAL 6,7-DISUBSTITUTED AND 7,8-DISUBSTITUTED 1-ALKYL-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXYLIC ACIDS [J].

KOGA, H ;

ITOH, A ;

MURAYAMA, S ;

SUZUE, S ;

IRIKURA, T .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (12) :1358-1363

[7]

MATSUMOTO H, 1982, Patent No. 72981

[8] PYRIDONE-CARBOXYLIC ACID ANTIBACTERIAL AGENTS .3. SYNTHESIS OF FLUORINATED PYRIDINES BY THE BALZ-SCHIEMANN REACTION - AN ALTERNATIVE ROUTE TO ENOXACIN, A NEW ANTIBACTERIAL PYRIDONECARBOXYLIC ACID [J].

MATSUMOTO, J ;

MIYAMOTO, T ;

MINAMIDA, A ;

NISHIMURA, Y ;

EGAWA, H ;

NISHIMURA, H .

JOURNAL OF HETEROCYCLIC CHEMISTRY, 1984, 21 (03) :673-679

[9] PYRIDONECARBOXYLIC ACIDS AS ANTIBACTERIAL AGENTS .2. SYNTHESIS AND STRUCTURE ACTIVITY RELATIONSHIPS OF 1,6,7-TRISUBSTITUTED 1,4-DIHYDRO-4-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACIDS, INCLUDING ENOXACIN, A NEW ANTIBACTERIAL AGENT [J].

MATSUMOTO, J ;

MIYAMOTO, T ;

MINAMIDA, A ;

NISHIMURA, Y ;

EGAWA, H ;

NISHIMURA, H .

JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (03) :292-301

[10]

REED L. J., 1938, AMER JOUR HYG, V27, P493

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