POTENTIAL MECHANISM-BASED INHIBITORS OF PROTEOLYTIC-ENZYMES

被引：15

作者：

GROUTAS, WC

BRUBAKER, MJ

VENKATARAMAN, R

EPP, JB

HOUSERARCHIELD, N

CHONG, LS

MCCLENAHAN, JJ

机构：

[1] Department of Chemistry Wichita State University Wichita

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1992年 / 2卷 / 02期

关键词：

D O I：

10.1016/S0960-894X(01)80445-5

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The design, synthesis, and inhibitory activity toward human neutropil elastase, of a series of potential mechanims-based inhibitors is described.

引用

页码：175 / 180

页数：6

共 18 条

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