AN EVALUATION OF TAMOXIFEN AS A PARTIAL AGONIST BY CLASSICAL RECEPTOR THEORY - AN EXPLANATION OF THE DUAL ACTION OF TAMOXIFEN

被引:36
作者
MACNAB, MW [1 ]
TALLARIDA, RJ [1 ]
JOSEPH, R [1 ]
机构
[1] TEMPLE UNIV,HLTH SCI CTR,SCH MED,DEPT PHARMACOL,PHILADELPHIA,PA 19140
关键词
D O I
10.1016/0014-2999(84)90493-X
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:321 / 326
页数:6
相关论文
共 25 条
[1]  
ARIENS EJ, 1954, ARCH INT PHARMACOD T, V99, P32
[2]  
Ariens EJ., 1964, MOL PHARM
[3]  
BIANCO AR, 1982, REV ENDOCRINE RELA S, V9, P215
[4]  
BORGNA JL, 1981, J BIOL CHEM, V256, P859
[5]  
Clark A. J., 1937, HDB EXPERIMENTAL PHA, V4, P1
[6]   The reaction between acetyl choline and muscle cells. [J].
Clark, AJC .
JOURNAL OF PHYSIOLOGY-LONDON, 1926, 61 (04) :530-546
[7]   ESTROGEN-LIKE EFFECT OF TAMOXIFEN ON VAGINAL EPITHELIUM [J].
FERRAZZI, E ;
CARTEI, G ;
MATTARAZZO, R ;
FIORENTINO, M .
BRITISH MEDICAL JOURNAL, 1977, 1 (6072) :1351-1352
[8]  
GADDUM JH, 1937, J PHYSIOL-LONDON, V89, pP7
[9]   EFFECT OF ANTI-OESTROGEN TAMOXIFEN ON PLASMA-LEVELS OF LUTEINIZING-HORMONE, FOLLICLE-STIMULATING-HORMONE, PROLACTIN, ESTRADIOL AND PROGESTERONE IN NORMAL PREMENOPAUSAL WOMEN [J].
GROOM, GV ;
GRIFFITHS, K .
JOURNAL OF ENDOCRINOLOGY, 1976, 70 (03) :421-428
[10]  
HARPER MJK, 1967, J REPROD FERTIL, V13, P101