MEASUREMENTS OF CA-45-2+ UPTAKE AND CONTRACTILE RESPONSES AFTER ACTIVATION OF POSTSYNAPTIC ALPHA-1-ADRENOCEPTORS IN THE ISOLATED CANINE SAPHENOUS-VEIN - EFFECTS OF CALCIUM ENTRY BLOCKADE

被引:31
作者
JIM, KF [1 ]
DEMARINIS, RM [1 ]
MATTHEWS, WD [1 ]
机构
[1] SK&F LABS,DEPT MED CHEM,PHILADELPHIA,PA 19101
关键词
D O I
10.1016/0014-2999(85)90059-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:199 / 208
页数:10
相关论文
共 39 条
[1]  
AWAD R, 1983, J PHARMACOL EXP THER, V227, P60
[2]   FUNCTIONAL BASIS FOR CLASSIFICATION OF ALPHA-ADRENERGIC RECEPTORS [J].
BERTHELSEN, S ;
PETTINGER, WA .
LIFE SCIENCES, 1977, 21 (05) :595-606
[3]   CALCIUM ENTRY BLOCKING-DRUGS, CALCIUM-ANTAGONISTS AND VASCULAR SMOOTH-MUSCLE FUNCTION [J].
BOU, J ;
LLENAS, J ;
MASSINGHAM, R .
JOURNAL OF AUTONOMIC PHARMACOLOGY, 1983, 3 (03) :219-232
[4]   SODIUM-CALCIUM SITES IN SMOOTH-MUSCLE AND THEIR ACCESSIBILITY TO LANTHANUM [J].
BURTON, J ;
GODFRAIND, T .
JOURNAL OF PHYSIOLOGY-LONDON, 1974, 241 (02) :287-298
[5]   ALPHA-1-ADRENOCEPTORS INDUCE CA INFLUX AND INTRACELLULAR CA RELEASE IN ISOLATED RABBIT AORTA [J].
CAUVIN, C ;
LOUTZENHISER, R ;
HWANG, O ;
VANBREEMEN, C .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 84 (3-4) :233-235
[6]   L-1,2,3,4-TETRAHYDRO-8-METHOXY-5-(METHYLTHIO)-2-NAPHTHALENAMINE - A POTENT AND SELECTIVE AGONIST AT ALPHA-1-ADRENOCEPTORS [J].
DEMARINIS, RM ;
HIEBLE, JP .
JOURNAL OF MEDICINAL CHEMISTRY, 1983, 26 (09) :1215-1218
[7]   ALPHA-ADRENERGIC AGENTS .2. SYNTHESIS AND ALPHA-1-AGONIST ACTIVITY OF 2-AMINOTETRALINS [J].
DEMARINIS, RM ;
SHAH, DH ;
HALL, RF ;
HIEBLE, JP ;
PENDLETON, RG .
JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (02) :136-141
[8]  
DEMARINIS RM, 1984, J MED CHEM
[9]   UNEVEN DISTRIBUTION OF POSTJUNCTIONAL ALPHA-1-LIKE AND ALPHA-2-LIKE ADRENOCEPTORS IN CANINE ARTERIAL AND VENOUS SMOOTH-MUSCLE [J].
DEMEY, J ;
VANHOUTTE, PM .
CIRCULATION RESEARCH, 1981, 48 (06) :875-884
[10]   EFFECT OF LANTHANUM AND REDUCED TEMPERATURE ON CA-45 EFFLUX FROM RABBIT AORTA [J].
DETH, RC .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 234 (05) :C139-C145