CONFORMATIONAL-ANALYSIS OF THE DOPAMINE-RECEPTOR AGONIST "5-HYDROXY-2-(DIPROPYLAMINO)TETRALIN AND ITS C(2)-METHYL-SUBSTITUTED DERIVATIVE

被引：28

作者：

KARLEN, A

JOHANSSON, AM

KENNE, L

ARVIDSSON, LE

HACKSELL, U

机构：

[1] UNIV UPPSALA,UPPSALA BIOMED CTR,DEPT ORGAN PHARMACEUT CHEM,S-75123 UPPSALA,SWEDEN

[2] KABIVITRUM,DEPT ANALYT CHEM,S-11287 STOCKHOLM,SWEDEN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 06期

关键词：

D O I：

10.1021/jm00156a008

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：917 / 924

页数：8

共 42 条

[1]

Allinger N. L., 1980, QCPE, P395

[2] CONFORMATIONAL-ANALYSIS .130. MM2 - HYDROCARBON FORCE-FIELD UTILIZING V1 AND V2 TORSIONAL TERMS [J].

ALLINGER, NL .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1977, 99 (25) :8127-8134

[3] SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF SULFONIUM ANALOGS OF DOPAMINE - NON-CLASSICAL DOPAMINE AGONISTS [J].

ANDERSON, K ;

KURUVILLA, A ;

URETSKY, N ;

MILLER, DD .

JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (06) :683-687

[4]

ANDERSSON B, 1985, ACTA PHARM SUEC S, V2, P139

[5]

ARVIDSSON LE, 1981, J MED CHEM, V24, P923

[6]

BUCOURT R, 1974, TOP STEREOCHEM, V8, P159

[7]

CAMERMAN N, 1979, MOL PHARMACOL, V16, P729

[8] STRUCTURE-ACTIVITY-RELATIONSHIPS OF DOPAMINE AGONISTS [J].

CANNON, JG .

ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1983, 23 :103-130

[9]

CANNON JG, 1984, CRC HDB STEREOISOMER, P117

[10] CONFORMATIONAL REQUIREMENTS FOR NOREPINEPHRINE UPTAKE INHIBITION BY PHENETHYLAMINES IN BRAIN SYNAPTOSOMES - EFFECTS OF ALPHA-ALKYL SUBSTITUTION [J].

DEJONG, AP ;

FESIK, SW ;

MAKRIYANNIS, A .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (12) :1438-1441

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